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N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-3-(1-methyl-1H-pyrazol-4-yl)propanamide
(1R,7S)-N-methyl-4-oxo-3-[2-(piperidin-1-yl)ethyl]-N-[2-(1H-pyrazol-1-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(3R,7S,8aS)-7-{[(3-fluorophenyl)methyl]amino}-3-(hydroxymethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
3-(1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidin-3-yl)benzoic acid
N-(1-ethyl-4-methyl-1H-pyrazol-5-yl)-2-[5-(1-phenylcyclopropyl)-2H-1,2,3,4-tetrazol-2-yl]acetamide
(1R,5S,6S)-3-{[2-(furan-2-yl)phenyl]methyl}-6-(morpholine-4-carbonyl)-3-azabicyclo[3.1.0]hexane
2-[(4-phenylpiperidin-1-yl)methyl]-4-(pyrimidin-2-yl)phenol
6-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidin-3-yl)propanamide
1-phenyl-N-[1-(pyrazin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-1-[3-(methylsulfanyl)phenyl]urea
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]piperidin-4-ol
2-(3-fluorophenoxy)-1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]ethan-1-one
2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-4-[(4-methyl-1H-pyrazol-1-yl)methyl]-1,3-oxazole
2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]acetamide
methyl 1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylate
2-(3-fluorophenoxymethyl)-N-[(3-methylpyridin-4-yl)methyl]-1,3-oxazole-4-carboxamide
9-(1H-1,2,3-benzotriazole-5-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-1-azabicyclo[2.2.2]octan-3-amine
[(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl][(2E)-3-(furan-2-yl)prop-2-en-1-yl]methylamine
1-({5-[1-(3-fluoropyridin-4-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)-4-methylpiperazine
9-(1H-1,2,3-benzotriazole-5-carbonyl)-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
(3S,7S,8aS)-7-{[(5-chlorothiophen-2-yl)methyl]amino}-3-[(4-hydroxyphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-({2-[1-(3-methoxybenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
{[5-(furan-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}(methyl)(thiophen-2-ylmethyl)amine
(3aR,5R,6S,7aS)-2-[2-(morpholin-4-yl)benzoyl]-octahydro-1H-isoindole-5,6-diol
2-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)acetamide
(3R,4S)-1-{[4-(methoxymethyl)piperidin-1-yl]sulfonyl}-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-1-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-(2-{1-[4-(4-fluorophenyl)-4-oxobutanoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
(2S,4S)-4-cyclopentaneamido-N-ethyl-1-(pyridine-3-carbonyl)pyrrolidine-2-carboxamide
2-[3-(dimethylamino)propyl]-9-(4-ethylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(1-benzylpiperidin-4-yl)methyl]-2-ethyl-N-methylpyridine-4-carboxamide
7-methyl-3-{[(prop-2-en-1-yl)(pyridin-2-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
6-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-3-carbonitrile
2-{[(3R,4S)-1-(2-methanesulfonylethyl)-4-propylpyrrolidin-3-yl]amino}pyridine-3-carbonitrile
2-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)quinolin-8-ol
8-(5-chloro-6-hydroxy-2-methylpyrimidin-4-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
ethyl 4-[2-(1H-pyrazol-1-yl)acetamido]piperidine-1-carboxylate
3-[(3-fluorophenyl)amino]-N-(4-methylphenyl)piperidine-1-carboxamide
8-{furo[3,2-c]pyridin-4-yl}-1-oxa-8-azaspiro[4.5]decane
3-({[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}(methyl)amino)-1λ6-thiolane-1,1-dione
3-[5-(ethoxymethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]-4-fluorobenzene-1-sulfonamide
1-(4-{[2-(4-chlorophenyl)ethyl]amino}-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-cyclobutanecarbonyl-N-[2-hydroxy-2-(pyridin-2-yl)ethyl]piperidine-4-carboxamide
4-[4-(1H-pyrazol-5-yl)benzoyl]thiomorpholine
6-methyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-(1H-1,2,4-triazol-1-yl)propan-1-one
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-2,3,5,6-tetramethylbenzamide
(1R,3R)-N1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}cyclopentane-1,3-diamine