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N-butyl-N-methyl-3-({methyl[2-(4-methylphenoxy)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
N5-(cyclohexylmethyl)-1-cyclopropyl-N3-(2-hydroxy-2-phenylethyl)-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]pyrrolidin-2-one
N-{[7-(1-benzothiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-3-fluorobenzamide
[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl})methylamine
5-(3,3-diphenylpiperidine-1-carbonyl)-3,4-dihydropyrimidin-4-one
N-cyclopropyl-1-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}piperidine-3-carboxamide
1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-4-[(4-fluorophenyl)methyl]piperidine
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
6-methoxy-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(3S,4S)-1-(2-hydroxyacetyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-(benzylamino)-1-{2-[2-(dimethylamino)ethyl]piperidin-1-yl}ethan-1-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)-N-propylacetamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(3-methylthiophene-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
N-butyl-N-(thiophen-3-ylmethyl)-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
1-(3-cyanophenyl)-3-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]urea
N-[(2R,3R)-2-methoxy-1'-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanamide
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-4-methylphenyl)urea
4-[(2-fluorophenyl)methyl]-1-(2-methoxy-2-phenylacetyl)-1,4-diazepan-5-one
(3S,4S)-4-(dimethylamino)-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]pyrrolidin-3-ol
1-(4-chloro-3-fluorophenyl)-3-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]urea
N-[(4-methoxyphenyl)methyl]-2-methyl-N-(2-methylpropyl)pyridine-3-carboxamide
3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]adamantan-1-amine
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5-{methyl[1-(1,3-thiazol-2-yl)ethyl]amino}azepan-2-one
6-{[5-(2-fluorophenyl)-1,2,4-triazin-3-yl]amino}-2-methylheptan-2-ol
4-(1H-imidazol-1-yl)-1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidine-4-carboxylic acid
2-{[4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazin-1-yl]methyl}benzonitrile
4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-N-(2-methoxypyridin-3-yl)benzamide
4-{[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]sulfonyl}-1-methyl-1H-imidazole
N-[(8-methoxyquinolin-5-yl)methyl]-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(2R,3R,6R)-3-phenyl-5-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
N-ethyl-2-fluoro-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)benzamide
4-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-N-methyl-1,3-thiazol-2-amine
(3S,5R)-1-cyclopropanecarbonyl-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[1-(propan-2-yl)piperidin-4-yl]pyridin-2-amine
N-methyl-2-[(prop-2-en-1-yl)amino]-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
2-(4-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)pyrazine
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-4-propylpyrimidine-5-carboxamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]propanamide
methyl (2S,4S)-1-methyl-4-{[(3-phenoxyphenyl)carbamoyl]amino}pyrrolidine-2-carboxylate
5-fluoro-2-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
2-{4-[(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
(1R,3S)-7-(2-aminopyridine-4-carbonyl)-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[1-(1H-imidazol-1-yl)ethyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
5-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyridine-2-carbonitrile
3-(furan-2-yl)-2-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]formamido}propanoic acid
(3S,4S)-1-methanesulfonyl-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid