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methyl({1-[1-(2-phenylbenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)amine
3-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-N-(5-methyl-1,3-thiazol-2-yl)benzamide
N-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-2,3-dimethylquinoxaline-6-carboxamide
1-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-methyl-7-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
methyl 2-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-1,3-oxazole-4-carboxylate
1-{4-[2-(3-methoxypropyl)piperidine-1-carbonyl]phenyl}-4-methylpiperazine
(4aS,8aR)-1-(2-methylpropyl)-6-(1H-pyrazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-(oxolan-2-ylmethyl)-3-(2-oxopyrrolidin-1-yl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzamide
9-(3-hydroxybenzoyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-(pyridin-4-yl)propanamide
2-(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]acetamide
1-(5-ethyl-2-methylpyrimidin-4-yl)-N-[3-(4-fluorophenyl)propyl]piperidin-4-amine
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-1,5-dimethyl-1H-pyrazole-3-carboxamide
2-({[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}amino)-2-methylpropan-1-ol
2-methoxy-1-[1'-(5-methyl-1,2-oxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
9-(3-ethyl-1H-pyrazole-5-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{5-[(3,4-dimethoxyphenyl)methyl]-1,3,4-thiadiazol-2-yl}-1-(piperidin-3-yl)urea
1-[2-(dimethylamino)-6-(2,2-dimethylpropyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
N-cyclopentyl-3-{[(2-fluoro-5-methoxyphenyl)methyl]amino}-5-(phenylsulfamoyl)benzamide
[(2,2-dimethyl-1-phenylcyclopropyl)methyl](methyl){[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
5-chloro-2-[2-(pyridin-3-yl)-1H-imidazol-1-yl]pyridine
N-methyl-3-propyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
6-{3-hydroxy-5-[2-(piperidin-2-yl)ethyl]phenyl}-2H-1,3-benzodioxole-5-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-3-(propan-2-yl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-6-[(2-phenyl-1,3-thiazol-5-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-{[3-(2,6-dimethylphenoxy)azetidin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
1-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
3,5-difluoro-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyridine-2-carboxamide
2-{3-[(1-methylpiperidin-4-yl)methyl]-5-[2-(2-oxoazepan-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
3-{[(5-ethylfuran-2-yl)methyl]amino}-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-5-[(propan-2-yl)sulfamoyl]benzamide
N-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)[1-(pyridin-3-yl)ethyl]amine
1-(4-chloro-2-methoxybenzoyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
2-{2-[(1,1-dioxo-1λ6-thian-3-yl)methyl]phenoxy}-N-methylacetamide
2-{[1-(2-fluorophenyl)-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]methyl}morpholine
1-(2-methanesulfonylethyl)-5-(6-methyl-2H-1,3-benzodioxol-5-yl)-4-phenyl-1H-imidazole
(3R,5S)-N-[3-(morpholin-4-yl)propyl]-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
1-[2-(dimethylamino)ethyl]-5-(oxolane-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamide
8-methoxy-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[2-(dimethylamino)-4-[(pyridin-3-ylmethyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-(4-fluorophenyl)-4-(1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)piperazine
2-(2-{2,5-dimethyl-3-[(3-methylpiperidin-1-yl)methyl]phenyl}-1H-imidazol-1-yl)ethan-1-ol
2-ethyl-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}benzamide
8-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
(5S,9aS,9bS)-5-(2,1,3-benzoxadiazol-5-yl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidine-1-carbonyl]benzene-1-sulfonamide
2-{1-ethyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-(quinoxalin-6-ylmethyl)acetamide
5-ethyl-N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine