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N-[(3S,4R)-4-(4-methoxyphenyl)-1-(4-methylpyridine-3-carbonyl)pyrrolidin-3-yl]acetamide
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl){2-phenyl-1-[1-(1-phenyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]ethyl}amine
4-{4-[(3-methylthiophen-2-yl)methyl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-methyl-6-(propan-2-yl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]pyrimidin-4-amine
3-{5-[1-(pyridine-4-carbonyl)piperidin-4-yl]-1,2,4-oxadiazol-3-yl}pyridazine
(3aR,7aS)-2-(4-phenyl-1H-imidazole-5-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-[(1-cyclopentylpiperidin-3-yl)methyl]-N-[2-(piperidin-1-yl)ethyl]cyclopropanecarboxamide
5-(1-butanoylpiperidin-4-yl)-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(3-methoxyphenyl)methyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-(2-methylpropyl)acetamide
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(pyrimidin-2-ylsulfanyl)acetamide
1-[3-({[(2-fluorophenyl)methyl](methyl)amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
3-(2,6-diethylphenyl)-1-{[4-(hydroxymethyl)oxan-4-yl]methyl}-1-methylurea
2-(3-fluorophenyl)-1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-benzoyl-1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
4-(3-hydroxypyrrolidine-1-carbonyl)-N-(1H-imidazol-2-ylmethyl)benzene-1-sulfonamide
2-[(4-chlorophenyl)methyl]-N-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
2-methyl-8-(2-methyl-1,8-naphthyridine-3-carbonyl)-2,8-diazaspiro[4.5]decane
(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-N-(2-hydroxypyridin-3-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide
N-[(2S)-1-hydroxy-3-methylbutan-2-yl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
5-[2-(1-benzofuran-5-yl)-1H-imidazol-1-yl]-2-hydroxy-N,N-dimethylbenzamide
N-cyclopropyl-6-(4-methoxy-2-methylphenyl)pyridazin-3-amine
3-hydroxy-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2-methylbenzamide
(3aR,6aR)-2-(cyclobutylmethyl)-5-[2-(3,4-difluorophenyl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-(2-hydroxyethyl)-2-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
3-(1H-imidazol-1-yl)-5-(morpholine-4-sulfonyl)benzoic acid
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[4-(methylsulfanyl)phenyl]acetamide
2-[4-(5-chloropyridine-2-carbonyl)morpholin-3-yl]-N-(2,2,2-trifluoroethyl)acetamide
2-(propan-2-ylsulfanyl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1-(pyridin-2-ylmethyl)piperidin-2-one
N-(1-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-fluorobenzamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
N-methyl-2-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
1'-(2,3-dihydro-1H-inden-2-yl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
6-[3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-2-carbonitrile
1-(2-methoxyphenyl)-3-{1-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
4-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}benzoic acid
5-ethyl-4-[4-(4-fluorophenoxy)piperidin-1-yl]pyrimidin-2-amine
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}pyridine-3-carboxamide
N-cyclohexyl-1-{1,3-dioxo-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-3-carboxamide
3-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
6-chloro-1-methyl-N-[2-(2-methylpropanesulfonyl)ethyl]-1H-indole-2-carboxamide
N-(2-{[3,5-dichloro-4-(prop-2-en-1-yloxy)phenyl]formamido}ethyl)acetamide
N,2-dimethyl-N-[2-(oxan-4-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
4-{[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2,1,3-benzoxadiazole
1-(1-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
methyl 2-[(4aS,8aR)-decahydroisoquinoline-2-sulfonyl]-6-(pyridin-3-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate