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3-(2-ethyl-1H-imidazol-1-yl)-1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}propan-1-one
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(5-methyl-1H-pyrazole-3-carbonyl)piperidin-3-ol
2-(1,3-benzoxazol-2-yl)-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]acetamide
N-[(2-chlorophenyl)methyl]-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(4-methyl-1H-pyrazol-1-yl)propanamide
3-{[1-(2-cyclohexyl-1H-imidazol-1-yl)propan-2-yl]oxy}pyridine
4-[(4-methyl-1H-imidazol-5-yl)methyl]-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
(2S)-N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-hydroxypropanamide
3-(1-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-3-yl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1-methyl-1H-indazol-6-yl)-4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carboxamide
3-butyl-1-{2-[2-(furan-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(pyridin-3-yl)-3-(thiophen-3-yl)propanamide
1-[(3-methylpyridin-2-yl)methyl]-4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine
N-(2-hydroxyethyl)-1-methyl-N-[(2-methylphenyl)methyl]-5-phenyl-1H-pyrrole-2-carboxamide
4-{[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1-methyl-1H-pyrazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(4-chlorophenyl)methyl]-N-[(3-fluoro-4-methylphenyl)methyl]-6-oxopiperidine-3-carboxamide
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-(4,4,4-trifluorobutyl)piperidin-4-ol
(1R,2R,6S,7S)-4-[4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carbonyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
methyl 2-[(cyclohexylmethyl)sulfamoyl]-6-(4-hydroxy-4-methylpentan-2-yl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-cyclopropanecarbonyl-1'-(3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-cyclopropyl-8-{[4-(1H-imidazol-1-yl)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
2-{4-[6-amino-5-cyano-4-(3-ethyl-1,2-oxazol-5-yl)pyridin-2-yl]phenoxy}acetic acid
3-[3-(cyclopropylmethyl)-5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
2-{1-[(3-chloropyridin-4-yl)methyl]piperidin-4-yl}-1H-1,3-benzodiazole
N-(1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
N-{[3-(trifluoromethyl)phenyl]methyl}imidazo[1,2-a]pyridine-6-carboxamide
2-[methyl({2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl})amino]ethan-1-ol
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-[4-(hydroxymethyl)piperidin-1-yl]pyridine-3-carboxamide
N-cyclopropyl-5-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-cyclopropyl-5-(1H-indazole-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2,3-dimethyl-5-phenyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
3-(2H-1,3-benzodioxol-5-yl)-1-[3-(2-methoxybenzoyl)piperidin-1-yl]propan-1-one
(3R,5S)-N3-methyl-N3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N5-(6-methylpyridin-3-yl)piperidine-3,5-dicarboxamide
N-(3-phenylprop-2-yn-1-yl)-3-(propan-2-yl)-N-propyl-1,2-oxazole-5-carboxamide
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-[4-(4-methoxyphenoxy)piperidin-1-yl]propan-1-one
1-[(3-fluorophenyl)methyl]-5-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1H,4H-pyrazolo[3,4-d]imidazole
(4aR,7aS)-1-(cyclopropylmethyl)-4-(2,4-dimethylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-[2-(2,4-difluorophenoxy)propanoyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methyl-4-sulfamoylbenzamide
7-(pyridin-2-ylmethyl)-N-[2-(1H-1,2,3-triazol-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-(1H-1,3-benzodiazol-2-yl)-N-[(3-hydroxypyrrolidin-3-yl)methyl]propanamide
4-(pyridin-3-yl)-2-(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)pyrimidine
3-[({1-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}oxy)methyl]pyridine
(2R)-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-hydroxy-2-phenylacetamide
1-({3-methanesulfonylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)azepan-3-amine
8-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-[2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carbonyl]morpholine-2-carboxylic acid