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N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-1H-1,2,3-benzotriazole-5-carboxamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-(4-methyl-3-phenylpiperazin-1-yl)propan-1-one
N-(3-fluorophenyl)-2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholine-4-carboxamide
4-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
ethyl 4-({cyclopropyl[(5-methylthiophen-2-yl)methyl]carbamoyl}amino)benzoate
{[2-(furan-2-yl)pyrimidin-5-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(1-cyclobutanecarbonylpiperidin-3-yl)piperazine
N-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}pyrimidin-2-amine
N-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
3-({1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)pyridine
N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-4-(pyridin-2-yl)pyrimidin-2-amine
7-[5-(ethylsulfanyl)thiophene-2-carbonyl]-3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine
(3S,4S)-1-(benzenesulfonyl)-4-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}pyrrolidin-3-ol
2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-3-(piperidine-1-carbonyl)pyrazine
({5-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]furan-2-yl}methyl)dimethylamine
N-methyl-2-propyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1,3-thiazole-4-carboxamide
N-[(3R,4S)-1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-4-propylpyrrolidin-3-yl]cyclopropanesulfonamide
N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
N-[2-(morpholin-4-yl)ethyl]-4-{4-[(pyridin-2-ylmethyl)amino]piperidin-1-yl}benzamide
(2S,4S)-4-amino-1-[2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)acetyl]-N-methylpyrrolidine-2-carboxamide
5-(1H-imidazol-1-ylmethyl)-2-[2-(2-methylpropoxy)phenyl]pyridine
2-{[(2E)-3-phenylprop-2-en-1-yl]sulfanyl}-N-(pyrrolidin-3-yl)pyridine-3-carboxamide
3-(3,5-dimethylphenyl)-1-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]propan-1-one
1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-3-(N-methylmethanesulfonamido)propanamide
N-cycloheptylpiperidin-4-amine
N-(2,3-dimethylphenyl)-N'-[2-(4-hydroxyphenyl)ethyl]propanediamide
(3aS,6aS)-5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-cyclopropanecarbonyl-4-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecane
2-(pyridazine-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[(4-phenyloxan-4-yl)methyl]acetamide
ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})(quinolin-2-ylmethyl)amine
(2S,4R)-1-[(4-chlorophenyl)methyl]-4-{[(2,4-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
1-(4-{[(2-ethyl-2H-1,2,3,4-tetrazol-5-yl)amino]methyl}thiophen-2-yl)ethan-1-one
5-(azocane-1-carbonyl)-2-cyclopropyl-3,4-dihydropyrimidin-4-one
6-fluoro-N-[1-(morpholin-4-ylmethyl)cyclopentyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-chloro-N-(1-hydroxypropan-2-yl)-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
3-({1-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]pyrrolidin-3-yl}methyl)benzoic acid
1-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-(thian-4-yl)piperazine
1-(furan-3-carbonyl)-N-[2-(4-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(3-fluorophenyl)ethan-1-one
5-[(adamantan-2-ylmethyl)amino]-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-3-(thiophene-2-carbonyl)piperidine
5-({5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
dimethyl(2-{2-[6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazol-5-yl]-1H-imidazol-1-yl}ethyl)amine
4-(3,6-dimethylpyrazin-2-yl)-1-[(3-methylphenyl)methyl]piperazin-2-one
3-(3-chloro-2-fluorophenyl)-1-(1,4-dioxan-2-ylmethyl)-1-methylurea
4-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
1-{[2-(methylsulfanyl)phenyl]methyl}-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol