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6-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
4-(3-methylphenoxy)-1-(2-oxo-2,3-dihydro-1H-imidazole-4-carbonyl)piperidine-4-carboxylic acid
(benzylsulfamoyl)[2-(1H-indol-1-yl)ethyl]methylamine
1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
3-(5-aminopyrazin-2-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
1-methyl-4-{5-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-1-yl}piperidine
N-ethyl-1-[(2-methoxyphenyl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-oxopiperidine-3-carboxamide
1-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(pyridin-3-ylmethyl)piperazine
1-(4-phenyl-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidin-4-yl)ethan-1-one
1-(5-{[3-(3-chlorophenyl)pyrrolidin-1-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
N-[4-(furan-2-yl)butan-2-yl]-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
3-(1H-indazol-1-yl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
6-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
4-(2,6-dimethylpyridin-3-yl)-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]pyrimidin-2-amine
2-oxo-N-{2-[(pyridin-3-yl)amino]ethyl}-1-oxaspiro[4.5]decane-4-carboxamide
ethyl 4-(4-{4-[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]piperidin-1-yl}benzoyl)piperazine-1-carboxylate
2-amino-8-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
3-{2-[4-(2-phenylpropyl)-1H-1,2,3-triazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[1-(3,5-dimethyl-1H-indole-2-carbonyl)piperidin-4-yl]-N-phenylpropanamide
2-{2-[7-(dimethylamino)-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl]phenoxy}acetic acid
2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]{[(1R,5S,6R)-3-(morpholine-4-carbonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}amine
(3S,4R)-1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-phenylpyrrolidine-3-carboxylic acid
4-hydroxy-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-methylbenzamide
1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]-4-[(4-fluorophenyl)methyl]-1,4-diazepan-5-one
4-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
N-[(3S,4R)-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
1-[2-methoxy-5-({[2-(2-methylphenyl)ethyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
3-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-5-yl)-1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]urea
5-chloro-N-[1-(1H-imidazol-1-yl)butan-2-yl]pyridine-2-carboxamide
7-[4-(6-hydroxypyrimidin-4-yl)piperidine-1-carbonyl]-1,3-diazepane-2,4-dione
3-[1-(2,1-benzoxazole-3-carbonyl)piperidin-4-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl){[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}amine
N'-(adamantan-1-yl)-N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylpropanediamide
2-ethyl-9-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
7-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-5-propyl-1,2-oxazole-3-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}piperidin-2-one
5-(1H-imidazol-1-ylmethyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}furan-2-carboxamide
N-methyl-5-(1-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}pyrrolidin-2-yl)thiophene-2-carboxamide
(1R,5R)-6-(3-methoxybenzoyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-(4-ethoxy-3-methylphenyl)-N-(2-methanesulfonamidoethyl)butanamide
(2S,4S)-4-amino-1-(4-tert-butylbenzenesulfonyl)-N-ethylpyrrolidine-2-carboxamide
2-(3-phenylpropyl)-8-(1H-pyrazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(4aR,7aS)-1-(2-methoxyethyl)-4-[(6-methylpyridin-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[cyclohexyl(methyl)amino]-3-[2-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)phenoxy]propan-2-ol
ethyl 1-(2H-1,3-benzodioxole-5-carbonyl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
2-(furan-2-yl)-N-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine