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2-(2,3-dihydro-1H-inden-1-yl)-1-[4-(morpholine-4-carbonyl)piperazin-1-yl]ethan-1-one
(4aS,7aR)-1-(3-methylbenzoyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-3-yl)-4-phenylpiperazine
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-(pyrrolidin-1-yl)piperidin-3-yl]-1-[4-(3-methoxyphenyl)piperazin-1-yl]propan-1-one
2-[5-(1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
3-[(2R,3R,6R)-5-(1H-1,2,3-benzotriazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-cyclobutyl-3-[(2-methanesulfonamidoethyl)sulfamoyl]benzamide
2-{[(3S,4S)-3-hydroxy-4-(piperidin-1-yl)pyrrolidin-1-yl]methyl}-3,5-dimethoxybenzoic acid
N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-1-[(4-methylphenyl)amino]cyclopentane-1-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(1-propylpiperidin-4-yl)acetamide
dimethyl({2-[4-(quinolin-2-yl)morpholin-2-yl]ethyl})amine
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(thiolan-3-yl)piperidine
ethyl 4-(2-phenylethyl)-1-[2-(pyrimidin-2-ylsulfanyl)acetyl]piperidine-4-carboxylate
N-(1H-indol-3-yl)-6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-(4-acetylphenyl)-4-methylbenzamide
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(pyridin-2-yl)propan-1-one
5-[(benzyloxy)methyl]-1-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-phenyl-1H-imidazole
3-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-3-yl}-N-(2-fluorophenyl)propanamide
2-[5-(methoxymethyl)-1H-pyrazol-3-yl]-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-{[3-(azocane-1-carbonyl)-1,2-oxazol-5-yl]methoxy}-2-methyl-1,3-benzothiazole
2,6,8-trimethyl-4-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]quinoline
2-(4-{[2-(2-chloro-6-fluorophenyl)-1H-imidazol-1-yl]methyl}-1,3-thiazol-2-yl)pyrazine
3-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-6-methylpyridin-2-ol
N-methyl-N-(2-methylprop-2-en-1-yl)-3-propanamidobenzamide
7-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-(1H-1,3-benzodiazol-2-ylmethoxy)ethan-1-one
1-(1H-imidazol-4-ylmethyl)-4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-1,4-diazepan-6-ol
N-cyclopentyl-4-(4-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-ylmethyl}-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
1-{3-[4-(1,3-thiazol-2-yl)-1H-1,2,3-triazol-1-yl]propyl}-1H-indole
2-[5-cyclobutyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
1-[cyclohexyl(methyl)amino]-3-[4-({[2-(4-fluorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
2-(4-{[(3-methoxypropyl)(methyl)amino]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
2-[2-oxo-4-(4-oxo-1,4-dihydroquinoline-2-carbonyl)piperazin-1-yl]benzonitrile
ethyl 4-[4-(4-{[(3S)-2-oxoazepan-3-yl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
2-(2-tert-butylpyrimidin-5-yl)-N,6-dimethyl-N-(propan-2-yl)quinoline-4-carboxamide
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-methyl-2-(morpholine-4-carbonyl)-N-[2-(pyridin-2-yl)ethyl]pyridin-4-amine
methyl 3-[6-oxo-2-(pyrrolidin-1-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-8-yl]benzoate
N-(3-methoxyphenyl)-3-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}propanamide
4-(2-{2-[(4-ethoxypiperidin-1-yl)methyl]phenoxy}ethyl)morpholine
2-[({1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-3-yl}oxy)methyl]pyridine
4-(2H-1,3-benzodioxol-5-yl)-2-({[(1-hydroxycyclohexyl)methyl]amino}methyl)phenol
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]ethan-1-one
5-[2-(morpholin-4-ylmethyl)phenyl]-N-propylfuran-2-carboxamide
2-methyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-4,5,6,7-tetrahydro-1-benzofuran-4-one
3-methyl-5-{2-oxo-2-[3-(2-phenylacetyl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(6-fluoropyridin-3-yl)-3-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]urea
N-butyl-N-[(4-fluorophenyl)methyl]-2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]acetamide