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7-{[(furan-2-ylmethyl)(prop-2-en-1-yl)amino]methyl}-4-methyl-2H-chromen-2-one
5-{1-[2-(2,3-difluorophenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
2-(1,3-benzothiazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline
4-{[2-(dimethylamino)-2-(3-fluorophenyl)acetamido]methyl}benzoic acid
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-[4-(propan-2-yl)piperazin-1-yl]pyridine-3-carboxamide
6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridin-3-ol
1-[2-(cyclopent-2-en-1-yl)acetyl]-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
9-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-hydroxy-2,2-dimethyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-phenylpropanamide
3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidine
1-(5-tert-butyl-2-methoxyphenyl)-3-[(5-methyl-1H-imidazol-4-yl)methyl]urea
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-(hydroxymethyl)pyridine-2-carboxamide
5-(4-phenylazepane-1-carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(1-cyclopropanecarbonylpiperidine-4-carbonyl)-2-(1,3-thiazol-2-yl)piperidine
[3-(cyclopropylmethyl)-1-[3-(3-fluorophenyl)benzoyl]piperidin-3-yl]methanol
N-[1-(2,6-dimethylphenoxy)propan-2-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
7-(5-hydroxypyrazine-2-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(methylsulfanyl)-5-({3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)pyrimidine
1-(cyclohexylmethyl)-N-methyl-6-oxo-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-3-carboxamide
7-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-N,N,2-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-(3-methoxyphenyl)-3-[1-(oxolane-3-carbonyl)piperidin-4-yl]propanamide
1-(3-methoxy-4-methylphenyl)-3-[(3-methyloxetan-3-yl)methyl]urea
(3S,4R)-3-methoxy-1-(1,3,7-trimethyl-1H-indole-2-carbonyl)piperidin-4-amine
N,N-dimethyl-4-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]benzamide
3-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1-[(1R)-1-phenylethyl]urea
2-fluoro-5-sulfamoyl-N-(1,2,3,4-tetrahydronaphthalen-2-yl)benzamide
1-(1,3-benzothiazole-2-carbonyl)-1,4-diazepan-6-ol
2-amino-N-[(2,3-difluoro-4-methoxyphenyl)methyl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-1-(carbamoylmethyl)piperidine-4-carboxamide
2-(azepan-1-yl)-1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
6-methyl-2-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)quinolin-4-ol
1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
N-cyclopropyl-1-(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)piperidine-3-carboxamide
3-[(4-methoxyphenyl)methyl]-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethan-1-one
2-{4-[(3-ethoxyphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
N-[3-(1H-imidazol-1-yl)propyl]-5-[1-(pyridin-4-ylmethyl)pyrrolidin-2-yl]thiophene-2-carboxamide
2-(3-{[2-methyl-4-(2-methylphenyl)piperazin-1-yl]methyl}phenoxy)acetamide
5-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidine-1-carbonyl]pyrazin-2-ol
3-{3-[1-(dimethylamino)ethyl]phenyl}-4-methoxybenzoic acid
N,4-dimethyl-3-(2-oxoimidazolidin-1-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
8-({3-carboxypyrazolo[1,5-a]pyrimidin-6-yl}methyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-(4-chlorophenoxy)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylic acid
(3S)-1-(5-{2-azaspiro[4.4]nonane-2-carbonyl}-1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-3-ol
ethyl N-{[(2S,4S)-4-fluoro-1-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]pyrrolidin-2-yl]methyl}carbamate
3-methyl-7-[2-(thiophen-2-yl)azetidine-1-carbonyl]-3,4-dihydroquinazolin-4-one
(2S)-1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-N-[4-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
3-[(oxolan-3-ylmethyl)sulfamoyl]-N-(1,3-thiazol-2-ylmethyl)benzamide
3-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-4-(1H-1,2,4-triazol-5-yl)benzamide