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1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(1-methylpiperidin-4-yl)piperazine
(1R,5R)-6-(cyclopropylmethyl)-3-(5-fluoro-3-methyl-1H-indole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-methyl-4-({5-[1-(3-phenylpropyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
3-({[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
5-{[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
1-(1H-pyrrole-3-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-[(4-fluorophenyl)methyl]-N-[(2-methoxyphenyl)methyl]-2-(2-oxopiperidin-1-yl)acetamide
2-[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-2-(5-methyl-1,2-oxazol-3-yl)piperidine
7-(3,6-dimethylpyrazin-2-yl)-4-[2-(2-hydroxyethoxy)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(2,4-dimethylphenoxy)-3-{[1-(1-methylcyclopropyl)ethyl]amino}propan-2-ol
3-(pyridin-2-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
4-(5-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}pyrimidin-2-yl)morpholine
8-({3-[3-(benzyloxy)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)quinoline
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-2-(3-methoxypiperidin-1-yl)pyridine
4-(2-methoxyethyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-[1-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-1,3,4-thiadiazol-2-amine
9-[6-(dimethylamino)pyrazin-2-yl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2-(pyrrolidin-3-yl)benzamide
2-[({[4-(3-methoxyphenyl)-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]phenol
2-benzyl-8-{5-methyl-1-[4-(pyridin-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}-2,8-diazaspiro[5.5]undecane
1-[4-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,6-dimethyl-1-benzofuran-2-carboxamide
4-(2-fluoro-5-methylphenoxy)-1-(furan-2-carbonyl)piperidine-4-carboxylic acid
N-[3-(1H-pyrazol-1-yl)phenyl]-1-[3-(1H-pyrazol-1-yl)propanoyl]pyrrolidine-2-carboxamide
methyl 3-[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)carbamoyl]propanoate
3-amino-1-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
1-ethyl-4-{[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-3-methyl-1H-pyrazole
2-{4-[2-(2-methoxyethoxy)acetyl]-5-methyl-2-oxopiperazin-1-yl}benzonitrile
4-(1,2-oxazolidine-2-carbonyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine
2-[5-(cyclopent-1-en-1-ylmethyl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]acetic acid
1-(pyridin-3-ylmethyl)-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,4-diazepane
5-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrazin-2-ol
8-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-1-oxa-8-azaspiro[4.5]decane
5-methanesulfonyl-2-methyl-N-(oxolan-2-ylmethyl)pyrimidin-4-amine
1-(azocan-1-yl)-3-[2-methoxy-5-({[2-(3-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-(4,5-dimethyl-1H-imidazol-1-yl)-1-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]ethan-1-one
3-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
N-[(4-fluorophenyl)methyl]-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-(1-cyclobutanecarbonylpiperidin-4-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-[1-({1-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}methyl)-1H-pyrazol-5-yl]acetamide
2-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2,7-diazaspiro[4.5]decane
1-({5-[(benzyloxy)methyl]-1,2,4-oxadiazol-3-yl}methyl)-4-methylpiperazine
2-[5-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-3-yl]pyridine
N-[2-(1H-imidazol-1-yl)ethyl]-6-phenylpyridazin-3-amine
4-(2-hydroxypyridine-3-carbonyl)-1-(2-methylphenyl)piperazin-2-one
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-3-(2-methyl-1H-indol-1-yl)propanamide
2-[2-(trifluoromethoxy)phenyl]pyridine-3-carboxamide
N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(1H-pyrazol-3-ylmethyl)amine