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4-(1-benzothiophene-5-carbonyl)piperazin-2-one
N-[2-(dimethylamino)ethyl]-3-{1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperidin-4-yl}propanamide
N-cyclopropyl-1-[(1s,4s)-4-[(2E)-3-(4-methoxyphenyl)prop-2-enamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-methyl-4-{3-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]phenyl}butan-2-ol
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-4-(thiophene-2-carbonyl)piperazine
ethyl 4-{[(oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}-1H-pyrazole-3-carboxylate
N-[4-(1H-indol-2-yl)phenyl]-1-propylpiperidine-4-carboxamide
2-cyclopropanecarbonyl-8-(4-methylpyridine-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(aminomethyl)-4-(4-methoxy-2-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]thiophene-3-carboxamide
(2R)-2-amino-1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-3-methoxypropan-1-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(5-methyl-1H-pyrazol-1-yl)propanamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-6-(propan-2-yl)pyridazin-3-amine
1-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)-3-phenylpropan-2-ol
[3-(5-ethyl-1H-pyrrole-2-carbonyl)-9-(1H-imidazol-2-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
2-{1-[(1S)-1-cyclopropyl-2-methoxy-2-oxoethyl]-4-phenyl-1H-imidazol-5-yl}benzoic acid
3-{[(3,4-difluorophenyl)methyl]sulfamoyl}-N-(2-methoxyethyl)benzamide
(2-{[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)amino}ethyl)dimethylamine
4-{3-[1-(dimethylamino)ethyl]phenyl}-N,6-dimethylpyrimidin-2-amine
N-[(4-fluorophenyl)methyl]-2-methyl-N-(oxolan-2-ylmethyl)-1,3-thiazole-4-carboxamide
N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-4-(4H-1,2,4-triazol-4-yl)benzamide
2-(methoxymethyl)-5-[3-(pyridin-3-yl)propyl]-1,3-benzoxazole
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(3-methyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methanol
5-chloro-2-[4-(1-methylpiperidin-4-yl)piperazine-1-carbonyl]phenol
4-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-6-methylpyrimidin-2-amine
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-methoxypropan-1-one
2-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carboxamide
7-[2-(4-fluorophenyl)piperidine-1-carbonyl]-3-methyl-3,4-dihydroquinazolin-4-one
4-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-1-oxaspiro[4.4]nonan-2-one
N-[2-(pyridin-3-yloxy)ethyl]-3,4-dihydro-2H-1-benzopyran-2-carboxamide
N-[2-(4-sulfamoylphenyl)ethyl]oxolane-3-carboxamide
2-[(3-fluoro-4-methylphenyl)methyl]-N-[(3R,4R)-3-hydroxypiperidin-4-yl]benzamide
3-(1H-1,3-benzodiazol-2-yl)-N-[2-(propylsulfanyl)phenyl]azetidine-1-carboxamide
3-({2-[1-(5-ethylthiophene-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-(4-{[4-(5-methylfuran-2-yl)phenyl]methyl}-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl)ethan-1-ol
2-{[4-(2,3-dichlorophenyl)-1H-1,2,3-triazol-1-yl]methyl}pyridine
2-tert-butyl-N-[(2,3-dimethoxyphenyl)methyl]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-amine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carboxamide
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-4-(1H-pyrazol-4-yl)butan-1-one
1-{3-[(4-methoxypiperidin-1-yl)methyl]phenoxy}-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
diethyl[(2-ethyl-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}furan-3-yl)methyl]amine
N-[(3R,4S)-4-propyl-1-[3-(1H-pyrazol-1-yl)propyl]pyrrolidin-3-yl]methanesulfonamide
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-(1H-pyrazol-1-yl)butanamide
4-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidine-1-carbonyl]phenol
2-{5-[2-(3-chloro-1,2-oxazol-5-yl)ethyl]-3-cyclopropyl-1H-1,2,4-triazol-1-yl}-3-methylpyridine
4-[(3-chloro-4-methoxyphenyl)methyl]-3-ethyl-1-methylpiperazin-2-one
3-[2-(1-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)ethyl]phenol
3-{2-[2-(4-fluorophenyl)azetidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1-methyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]phenol