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3-{2-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}azetidin-3-ol
N-{[7-(1-benzofuran-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(morpholine-4-sulfonyl)pyrrolidin-3-amine
6-methoxy-3-({methyl[3-(oxolan-2-yl)propyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-(1-cyclopentyl-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl)ethan-1-ol
N-methyl-2-phenyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
3-[(3R,4S)-1-(isoquinoline-1-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
1,3,6-trimethyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{[2-(3,4-dimethoxyphenyl)-7-methylquinolin-3-yl]methyl}-1-methylpiperazin-2-one
3-[({1-[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]piperidin-4-yl}amino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]acetamide
N-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
4-({8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)benzoic acid
methyl({[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl})(quinolin-6-ylmethyl)amine
2-cycloheptyl-1-{4-[4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
{5-[(4-benzoylpiperazin-1-yl)methyl]furan-2-yl}methanol
6-methoxy-3-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-methyl-5-{2-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
1-methyl-4-(2-methyl-2-{3-methyl-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}propyl)piperazine
3-(4-methyl-1,3-thiazol-5-yl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]propanamide
4-(1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}pyrrolidin-3-yl)-1-(2-methylpropyl)piperidine
N4-[(1-methanesulfonylpiperidin-3-yl)methyl]-5,6,7,8-tetrahydroquinazoline-2,4-diamine
2-[1-({1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]pyridine
1-{[5-(methoxymethyl)furan-2-yl]methyl}-3-[4-(trifluoromethyl)benzoyl]piperidine
1-methyl-2-oxo-N-{1-phenyl-3,6-diazatricyclo[4.3.1.13,8]undecan-9-yl}-1,2-dihydropyridine-3-carboxamide
N-[(2-chloropyridin-3-yl)methyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-methylacetamide
4-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-4-oxobutane-1-sulfonamide
3-[5-(4-fluorophenyl)-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl]propanamide
dimethyl(2-{2-[1-(pyridazine-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(3-methylpyridin-4-yl)-1,4-diazepane
ethyl 1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
(4aS,7aR)-1-(3-phenyl-1H-pyrazole-4-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-1H-1,2,3-benzotriazole-5-carboxamide
3-(1,3-benzothiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-hydroxy-4-oxo-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
2-methyl-4-[4-({4-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)phenyl]butan-2-ol
N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-[(2-oxopyrrolidin-1-yl)methyl]piperidine-1-carboxamide
N-(2-hydroxyethyl)-1-(1-{[4-(2-methylphenyl)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
2-(4-fluoro-2-methoxyphenyl)pyridin-4-amine
8-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
8-(quinoline-3-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-[(3S,4S)-3,4-dihydroxypiperidin-1-yl]-N-(2,3-dimethylphenyl)-2-oxoacetamide
7-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-4H-chromen-4-one
3-(2-oxo-2,3-dihydro-1H-indol-5-yl)-1-[2-(3-phenylpyrrolidin-1-yl)ethyl]urea
6-(4-ethylphenyl)-3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}imidazo[2,1-b][1,3]thiazole
1-(1-{6-[3-(hydroxymethyl)phenyl]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
2-(pyridin-3-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(pyrrolidin-1-yl)acetamide
N-[(3-methoxyphenyl)methyl]-3-[1-(3-phenylprop-2-ynoyl)piperidin-3-yl]propanamide