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2-(2-hydroxyethyl)-9-[2-(4-hydroxyphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[2-(2-fluorophenyl)ethyl]-3-(3-hydroxypropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}pyridine-3-sulfonamide
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1H-pyrrole-2-carboxamide
1-(1-ethyl-1H-pyrazole-5-carbonyl)-3-(4-methylphenoxymethyl)piperidine
3-(2-methylphenyl)-1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidine
3-chloro-2-[3-(pyridin-3-yl)azetidin-1-yl]pyridine
2-ethyl-9-{2-[ethyl(methyl)amino]acetyl}-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-{[(2S,4S)-1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-4-fluoropyrrolidin-2-yl]methyl}butane-1-sulfonamide
N-[(2S,4R,6S)-2-benzyl-6-(4-acetamidophenyl)oxan-4-yl]acetamide
1-[2-({[2-(azocan-1-yl)pyridin-3-yl]methyl}amino)pyrimidin-4-yl]piperidin-3-ol
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-5-ethyl-1,3-oxazole-4-carboxamide
3-[1-(1-methyl-1H-indazole-3-carbonyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
1-[(3-chlorophenyl)methyl]-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
3-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1-[2-methoxy-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
6-ethoxy-3-{[2-(trifluoromethyl)morpholin-4-yl]methyl}-1,2-dihydroquinolin-2-one
4-[(2-chlorophenyl)methyl]-1-(2-methylbenzoyl)-1,4-diazepan-5-one
N-[4-(4-{[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]amino}piperidin-1-yl)phenyl]benzenesulfonamide
3-{[4-(3-chlorophenyl)-5-{[methyl(quinoxalin-6-ylmethyl)amino]methyl}-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
1-{2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-3-methylpiperidine
1-{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}-N,N-diethylpyrrolidin-3-amine
3-methoxy-2-[4-(2-methoxyethoxy)phenyl]-6-methylpyridine
ethyl 2-[4-(8-fluoroquinoline-2-carbonyl)morpholin-3-yl]acetate
5-[3-(3,5-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridin-2-amine
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]propan-1-one
(2R,3R)-3-methoxy-1'-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(4-fluorophenyl)-4-(5-fluoropyrimidin-2-yl)piperazine-2-carboxamide
4-benzyl-1-methyl-3-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N,N-dimethyl-6-{[1-(3-phenylpropyl)piperidin-3-yl]amino}pyridine-3-carboxamide
N-benzyl-1-[(2-chloro-4-fluorophenyl)methyl]-N-(cyclobutylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-[5-(methoxymethyl)furan-2-carbonyl]-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
3-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]phenol
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
(3aS,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-(3,3,3-trifluoropropanoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[4-(2-methoxyphenoxy)piperidin-1-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
4-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]benzene-1-sulfonamide
5-(4-chloro-1H-indazol-1-yl)thiophene-2-sulfonamide
2,3-dimethyl-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]quinoxaline-6-carboxamide
2-(2-chlorophenyl)-3-methyl-6-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-3H-imidazo[4,5-b]pyridine
6-{7-ethyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4,6-dimethyl-5-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,2,3,4-tetrahydropyrimidin-2-one
N,N-dimethyl-5-{1-[2-oxo-2-(thiophen-2-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
[(2,2-dimethyloxan-4-yl)methyl]({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
3-(oxolan-3-yl)-5-{1-[4-(propan-2-yloxy)phenyl]cyclopentyl}-1,2,4-oxadiazole
N-cycloheptyl-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-(2-fluorophenoxymethyl)-4-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1,3-oxazole
methyl 1-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-3-(2-methylpropyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-pyrrol-1-yl)propan-1-one
4-(piperidin-1-yl)-1-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]butan-1-one
2-[1-(2-chlorophenyl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)acetamide