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methyl 6-[(4-methoxy-3-methylphenyl)methyl]-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-[3-(benzyloxy)azetidine-1-carbonyl]-1-(propan-2-yl)piperidine
1-[2-({[2-(methylsulfanyl)pyrimidin-4-yl]amino}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one
(3S,4S)-4-(dimethylamino)-1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)pyrrolidin-3-ol
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(2,2,2-trifluoroethyl)piperidine-4-carboxamide
3,3-dimethyl-1-(2-oxo-2-{3-oxo-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-9-yl}ethyl)urea
1-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-phenylprop-2-yn-1-one
4-fluoro-N-({1-[3-(4-methoxyphenyl)propanoyl]piperidin-3-yl}methyl)benzamide
1-(4-ethoxy-2-fluorophenyl)-3-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]urea
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-(thiolan-3-yl)pyridin-2-amine
3-(2-methoxyethyl)-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine-3-carboxylic acid
2-(2,5-dioxoimidazolidin-1-yl)-N-methyl-N-(quinolin-2-ylmethyl)acetamide
4-(4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperazin-1-yl)quinazoline
N-[(6-hydroxypyrimidin-4-yl)methyl]-2-(4-methylphenyl)quinoline-4-carboxamide
2-{2-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-yl]-2-oxoethyl}-5,6-dimethoxy-1,2-dihydroisoquinolin-1-one
(4S)-3-(2-{4-[(methylsulfanyl)methyl]piperidin-1-yl}-2-oxoethyl)-4-phenyl-1,3-oxazolidin-2-one
methyl 2-(4-{3,9-diazaspiro[5.5]undecan-3-ylmethyl}phenoxy)acetate
(1-methyl-1H-imidazol-2-yl)({1-[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperidin-4-yl})methanol
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
1-{[2-(5-methylfuran-2-yl)phenyl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
5-ethyl-2,3-dimethyl-N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-cyclopentyl-N-(1,4-dioxan-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1,4-dithiepan-6-yl)piperidin-3-ol
ethyl 5-{[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]methyl}furan-2-carboxylate
N-methyl-N-[(3-{1-[2-(1H-pyrrol-1-yl)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}-1,2-oxazol-5-yl)methyl]acetamide
N-[(4-methoxyphenyl)methyl]-5-methyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
9-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-ethyl-N,5-dimethyl-1,2-oxazole-4-carboxamide
1-[(4-chlorophenyl)methyl]-N-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-3-amine
3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]propanamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-3-phenylprop-2-ynamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}acetamide
N-[3-(4-chloro-3-methylphenoxy)-2-hydroxypropyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
4-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-6-(morpholin-4-yl)pyrimidin-2-amine
8-[(2S)-2-hydroxypropanoyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
N-[2-(4-methylmorpholin-2-yl)ethyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
3-chloro-6-[2-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridazine
6-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
1-(4-{5-cyclopropyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperazin-1-yl)ethan-1-one
2-amino-7-(3-hydroxypyridine-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(3-chlorobenzoyl)-1-[(2,4,6-trimethoxyphenyl)methyl]piperidine
N-[2-(4-cycloheptylmorpholin-2-yl)ethyl]cyclopropanesulfonamide
N-(2-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]formamido}ethyl)pyridine-3-carboxamide
7-(3-chlorophenyl)-4-(5-methylpyridine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl (1R,3S,3aR,6aS)-3-(4-fluoro-3-methylphenyl)-1-(2-methoxy-2-oxoethyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-(2-chlorophenyl)-3-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)propan-1-one
5-(2-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amino}pyrimidin-4-yl)-2-ethoxybenzoic acid
2-{1-[2-(propane-2-sulfonyl)ethyl]-1H-imidazol-2-yl}benzoic acid