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6-[(4-methyl-1,4-diazepan-1-yl)methyl]-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
(2S,4R)-4-amino-1-[(2S)-2-acetamido-4-methylpentanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(1,2-oxazol-3-ylmethyl)-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
N-tert-butyl-3-[(2S)-2-hydroxy-2-phenylacetamido]-2-methylbenzamide
11-(3,5-dichloro-4-methylbenzoyl)-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
4-(2-fluoro-5-methylphenoxy)-1-(pyrazin-2-yl)piperidine-4-carboxylic acid
2-(3-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}phenoxy)acetamide
(2S)-3-(1H-indol-3-yl)-2-{[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}propanoic acid
4-oxo-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-3,4-dihydrophthalazine-1-carboxamide
N-(4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}phenyl)acetamide
(4aS,8aR)-6-(5-chloropyridine-2-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
6-methyl-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(pyrrolidin-1-yl)pyrimidin-4-amine
(3S,5R)-1-benzyl-N3-[2-(dimethylamino)ethyl]-N5-(4-fluorophenyl)piperidine-3,5-dicarboxamide
2-(3-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)-5-propylpyrimidine
2-[ethyl({[2-(prop-2-en-1-yloxy)phenyl]methyl})amino]acetic acid
2,2-dimethyl-1-[7-(1,2,3,4-tetrahydroquinoline-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]propan-1-one
1-{6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidin-4-yl}piperidin-4-ol
1-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(piperidin-1-yl)ethan-1-one
1-(4-{[(2R)-oxolan-2-ylmethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)-2-(pyrrolidin-1-yl)ethan-1-one
N-(isoquinolin-5-ylmethyl)-6-methoxy-N-methyl-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-[1-(2-ethoxyethyl)-4-phenyl-1H-imidazol-5-yl]quinolin-7-ol
methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)(thiophen-3-ylmethyl)amine
2-(4-chlorophenyl)-5,8-dimethoxy-3-(morpholin-4-ylmethyl)quinoline
3-(3-methoxypropyl)-N-(2-methylnaphthalen-1-yl)piperidine-1-carboxamide
3-({1-[2-(oxan-4-yl)acetyl]piperidin-4-yl}methyl)-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]acetamide
1-[(3,5-difluorophenyl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
[2-(1H-imidazol-4-yl)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
1-[7-(furan-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-N,N-dimethylpiperidin-3-amine
4-({4-[2-(3-methylpiperidin-1-yl)ethoxy]phenyl}methyl)morpholine
4-amino-2-(4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine-5-carbonitrile
6-[2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)ethyl]-2-methylpyrimidin-4-ol
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-5-methyl-6-(morpholine-4-carbonyl)thieno[2,3-d]pyrimidin-4-amine
(1R,5S)-6-[(4-fluoro-3-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-{4-[(2-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-N,N-dimethylaniline
ethyl 3-{[3-(2-{methyl[2-(pyridin-2-yl)ethyl]carbamoyl}ethyl)piperidine-1-carbonyl]amino}propanoate
N-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-3-(2,6-dimethylphenoxy)azetidine-1-carboxamide
1-{4-[4-(2-amino-6-ethyl-5-methylpyrimidin-4-yl)piperazin-1-yl]phenyl}ethan-1-one
2-amino-6-(propan-2-yl)-4-[3-(1H-pyrazol-1-ylmethyl)phenyl]pyridine-3-carbonitrile
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(3-phenylpropanoyl)piperidin-3-yl]propanoic acid
2-({[(3R,4R)-4-(hydroxymethyl)-1-[4-(pyrrolidin-1-yl)benzoyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
9-[3-(3-fluorophenyl)propanoyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-4-(1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-amine
4-ethoxy-N-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]pyrimidin-2-amine
1-{[5-(2H-1,3-benzodioxol-5-yl)-2-hydroxyphenyl]methyl}-N,N-diethylpiperidine-3-carboxamide
1-(3-methylpyridin-4-yl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-1,4-diazepane
N-cyclopentyl-3-{5-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[2-(dimethylamino)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]acetamide
1-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
5-oxo-N-[(1-propyl-1H-pyrazol-4-yl)methyl]-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide