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N-(carbamoylmethyl)-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(2S)-2-acetamido-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-(methylsulfanyl)butanamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(1H-indol-5-ylmethyl)pyrrolidin-3-yl]methanol
5-{[3-(3-methoxypropyl)piperidin-1-yl]methyl}-2-(thiophen-2-yl)pyrimidine
1-cyclopentyl-4-({[5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]amino}methyl)pyrrolidin-2-one
9-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
N-[(3R,5S)-1-cyclobutanecarbonyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1H-pyrrole-3-carboxamide
2-methyl-4-(4-{[3-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]methyl}phenyl)but-3-yn-2-ol
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-ethylbenzamide
7-[5-(4-chlorophenyl)-4-methyl-1H-pyrazole-3-carbonyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
ethyl 1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-(3-phenylpropyl)piperidine-3-carboxylate
3-[1-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]benzoic acid
N-[2-(5-methylthiophen-2-yl)ethyl]-4-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
N-[3-(piperidine-1-carbonyl)-5-[({[3-(trifluoromethyl)phenyl]methyl}amino)methyl]phenyl]methanesulfonamide
1-(furan-3-ylmethyl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine
2-[(4-aminopiperidin-1-yl)methyl]-6,8-dimethylquinolin-4-ol
[1-cyclopentanecarbonyl-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[(4-methyl-1,3-thiazol-2-yl)methyl]piperidin-4-ol
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-fluoro-2-methylphenyl)urea
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(3-phenylpropyl)piperidin-3-yl]propanoic acid
N-({5-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
4-(2,4-difluorophenyl)-3-(2-methylpropyl)-4H-1,2,4-triazole
4-(4-{[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]amino}piperidin-1-yl)-N-(pyridin-3-ylmethyl)benzamide
N-[2-(pyridin-3-yl)ethyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
5-cyclopropyl-4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1,3-oxazole
6-[2-(3-fluorophenyl)-3-oxopiperazine-1-carbonyl]-2-methyl-2,3,4,5-tetrahydropyridazin-3-one
2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
N-[4-(3-fluorophenyl)phenyl]-1-(1,3-thiazole-4-carbonyl)piperidine-3-carboxamide
1-(cyclohex-3-en-1-ylmethyl)-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
8-(6-ethylpyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
6-(3-fluoro-4-methoxyphenyl)-N,N-dimethylpyridine-2-carboxamide
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
2,6-diamino-4-(6-chloro-2-fluoro-3-methylphenyl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-(2-methylpropyl)piperidine
1-[2-(2-hydroxyethyl)piperidin-1-yl]-3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propan-1-one
2-(4-fluoro-3-methylphenyl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
2-{[1-(2,5-dimethylphenyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,4-dimethylpiperazine
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]ethane-1-sulfonamide
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(3-hydroxyphenyl)ethan-1-one
3-[3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-1-methyl-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]urea
1-(cyclopropylmethyl)-4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine
N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3-(4-methylphenyl)propanamide
methyl 4-{[3-(cyclopropylcarbamoyl)-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}benzoate
5-methyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1-benzofuran-2-carboxamide
4,6-dimethyl-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyridine-3-carbonitrile
8-[(5-ethylpyridin-2-yl)methyl]-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
4-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]-4H-1,2,4-triazole
2-{[(2-fluorophenyl)methyl](methyl)amino}-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
(1S,5R)-3-(pyrazin-2-yl)-6-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane