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(1R,7S)-3-(2-ethoxyethyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-methyl-5-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
[(3R,4R)-1-(furan-3-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-[cyclohexyl(thiophen-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(3R,4S)-4-(3-methoxyphenyl)-1-(quinoxalin-2-yl)pyrrolidin-3-amine
8-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(2-methoxy-2-methylpropyl)-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
N-(2,4-difluorophenyl)-4-(pyridin-3-ylmethoxy)piperidine-1-carboxamide
(2S)-4-methyl-2-[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]pentan-1-ol
1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2-benzyl-8-{[4-(1H-imidazol-1-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
3-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamido)-4-(2-methylpiperidin-1-yl)benzamide
[(1R,3S,3aS,6aR)-5-phenyl-3-[3-(prop-2-en-1-yloxy)phenyl]-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
6-methyl-2-{[2-(1-methyl-1H-pyrazol-3-yl)piperidin-1-yl]methyl}quinolin-4-ol
1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-4-(piperidine-1-carbonyl)piperidine
1-(1H-imidazol-4-ylmethyl)-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-hydroxy-N-[(1R,2S)-2-phenylcyclopropyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(pyrazin-2-yl)ethyl]acetamide
N-(2-hydroxyethyl)-N-methyl-1-(1-{[3-(2-methylphenyl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
6-chloro-N-[2-(dimethylamino)ethyl]-3-fluoro-N-(2-hydroxyethyl)imidazo[1,2-a]pyridine-2-carboxamide
2-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-5-methylimidazo[1,2-a]pyridine
4-(2,4-dimethoxyphenyl)-2-methyl-6-(propan-2-yl)pyrimidine
5-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-N-methylfuran-2-carboxamide
N-(2,2-dimethylpropyl)-4-methyl-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
8-[(2-chloro-6-fluorophenyl)methyl]-3-(2-methoxyethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-chloro-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-3,5-dimethyl-1-benzofuran-2-carboxamide
7-(4-fluorophenyl)-2-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
7-cyclopentyl-2-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
4-[1-(2,2-dimethylpropyl)piperidin-4-yl]thiomorpholine
1-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)urea
3-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-{[(butylcarbamoyl)methyl](methyl)amino}-2-[4-(propan-2-yloxy)phenyl]acetic acid
7-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-5-phenylpyrazolo[1,5-a]pyrimidine
1-[(2-{4-[(dimethylamino)methyl]thiophen-2-yl}-1H-imidazol-1-yl)methyl]cyclohexan-1-ol
2-{1-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]piperidin-4-yl}propan-2-ol
2-ethoxy-6-{[(1-hydroxybutan-2-yl)(thiophen-3-ylmethyl)amino]methyl}phenol
1-{2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-ethyl-N-(2-methylprop-2-en-1-yl)piperidine-4-carboxamide
2-[2-(3-methoxyphenoxy)ethyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-({7-[(4-methoxy-2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-2-carboxamide
diethyl({3-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
N-methyl-N-[(5-methylfuran-2-yl)methyl]-2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]acetamide
1-{2-[(2-cyclohexyl-1H-imidazol-1-yl)methyl]phenyl}-1H-1,2,4-triazole
N-cyclopentyl-N-[(3-methylthiophen-2-yl)methyl]-2-(pyrrolidin-1-yl)acetamide
3-[1-(propan-2-yloxy)ethyl]-4-propyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-5-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}furan-2-carboxamide
4-{[(3S,5R)-1-benzyl-5-(pyrrolidine-1-carbonyl)piperidin-3-yl]methyl}morpholine
1-(2-{[(6-methyl-2-phenylpyrimidin-4-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
4-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]-1-[(4-methylphenyl)methyl]piperazin-2-one
3-{[2-(methylsulfanyl)phenyl]methyl}-1λ6-thiane-1,1-dione
(3R,4S)-4-{4-[(4-methanesulfonylphenyl)methyl]-1,4-diazepan-1-yl}oxolan-3-ol