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[(1-cyclohexylpiperidin-3-yl)methyl][(1-ethyl-1H-pyrazol-4-yl)methyl](pyridin-3-ylmethyl)amine
N4-(1,4-dioxan-2-ylmethyl)-N4-methyl-6-(morpholin-4-yl)pyrimidine-2,4-diamine
2-(2,3-dihydro-1H-indene-5-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
3-{2-[1-(2-fluoro-6-methoxybenzoyl)piperidin-2-yl]ethyl}phenol
1-(3-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}phenyl)ethan-1-one
5-ethyl-2-{[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
2-(methylsulfanyl)-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
methyl 2-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
5-methyl-5-(4-methylpent-3-en-1-yl)-1-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}piperidin-2-one
N-[4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-4-(pyridin-2-yl)piperazine-1-carboxamide
2-(4-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenyl)-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]piperidin-4-amine
N-{5-[(E)-2-phenylethenyl]pyridin-2-yl}acetamide
2-(diethylamino)-N-{[2-(dimethylamino)pyridin-3-yl]methyl}acetamide
1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
N-[(2-aminopyridin-3-yl)methyl]-4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzamide
N-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-methylpropyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
2-[4-(1-benzothiophen-3-yl)-2-(pyrrolidin-1-ylmethyl)phenoxy]-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
4-{2-[1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)piperidin-2-yl]ethyl}phenol
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-hydroxypropan-1-one
1-[1-(oxane-4-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
8-(5-ethyl-1,2-oxazole-3-carbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{2-[(4aR,8aR)-6-(3-methylbutyl)-decahydro-1,6-naphthyridin-1-yl]-2-oxoethyl}-4-phenyl-1,2-dihydrophthalazin-1-one
1-({2-[2-(4-ethylpiperazin-1-yl)ethoxy]phenyl}methyl)pyrrolidin-3-amine
2-[5-(6-ethoxyquinolin-2-yl)-4-phenyl-1H-imidazol-1-yl]ethan-1-amine
2-methylpropyl (1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxylate
4-methoxy-3-[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]benzene-1-sulfonamide
3,3-dimethyl-1-{[5-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}urea
2-(2-{[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
methyl 2-[4-(2-fluoroethyl)-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl]acetate
1-(2-methoxybenzoyl)-4-[1-(methoxymethyl)cyclobutanecarbonyl]piperazine
3-[2-(3-hydroxy-4-methoxyphenyl)ethyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-(acetamidomethyl)benzoate
9-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
({2-[4-(1H-imidazol-1-yl)butoxy]phenyl}methyl)(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
7-[1-(2,3-dimethylphenyl)piperidin-4-yl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
6-methyl-1-[1-oxo-1-(piperidin-1-yl)propan-2-yl]-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
2-[2-oxo-2-(3-phenoxyazetidin-1-yl)ethyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
6-chloro-N-cyclopropyl-3-fluoro-N-[(trimethyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
N-{[1-(2-methylpropyl)piperidin-3-yl]methyl}-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
1-[3-(2-oxopyrrolidin-1-yl)propyl]-5-(4-propyl-1,4-diazepane-1-carbonyl)piperidin-2-one
2-(3-{[cyclohexyl(pyridin-2-ylmethyl)amino]methyl}phenyl)-6-methyl-3,4-dihydropyrimidin-4-one
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
methyl 5-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1H-pyrazole-3-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
4-[(2,5-dimethoxyphenyl)methyl]-2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-(propan-2-yl)-N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-(5-{[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
N-[(3R,5S)-1-benzyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
6-cyclopentyl-N-(3-methoxy-2,2-dimethylpropyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine