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N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
4-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}-N-(3-methylpyridin-2-yl)benzamide
2-(piperidin-1-yl)-5-{[4-(thian-4-yl)piperazin-1-yl]methyl}pyrimidine
(2R,3R,6R)-5-[(3,4-difluorophenyl)methyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2S,4S)-1-cyclobutanecarbonyl-N-ethyl-4-(5-methoxyfuran-2-amido)pyrrolidine-2-carboxamide
6,6-dimethyl-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-5-oxothiomorpholine-3-carboxamide
1-(3-phenylpropyl)-4-(piperidin-3-ylmethyl)-1,4-diazepane
N-[3-(1H-pyrazol-1-yl)propyl]-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-1,2,3-thiadiazole-4-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-[(2-methyl-1,3-oxazol-4-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-ethyl-9-(1-methyl-1H-pyrazole-4-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
8-pentanoyl-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2-fluorophenoxymethyl)-N-[2-(pyrazin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
3-cyclopropyl-5-{[3-(thiophen-3-yl)-1H-pyrazol-1-yl]methyl}-1,2,4-oxadiazole
3-[4-(2-phenylethyl)piperazine-1-carbonyl]-5,6,7,8-tetrahydroquinoline
6-[4-(benzyloxy)piperidin-1-yl]pyridine-2-carboxylic acid
3-[(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}furan-2-yl)sulfanyl]-4-methyl-4H-1,2,4-triazole
8-[2-amino-6-(thiophen-2-ylsulfanyl)pyrimidin-4-yl]-2,8-diazaspiro[4.5]decan-3-one
7-(thiophen-2-yl)-4-{[3-(trifluoromethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-{furo[3,2-c]pyridin-4-yl}piperazine
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-(3-phenoxyazetidin-1-yl)ethan-1-one
N-(5-oxo-1-propylpyrrolidin-3-yl)-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
2-(3-{[4-(benzyloxy)piperidin-1-yl]methyl}phenyl)ethan-1-amine
1-({5-[1-(2H-1,3-benzodioxol-5-yl)-1H-1,2,4-triazol-5-yl]furan-2-yl}methyl)-4-methylpiperazine
N3-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-N5-[2-(pyridin-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
[(3-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)methyl](methyl)(pyridin-3-ylmethyl)amine
4-(2-methylphenoxy)-1-[3-(methylsulfanyl)propanoyl]piperidine-4-carboxylic acid
2-[1-(3,6-dimethylpyrazin-2-yl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-N,N-dimethylazepan-4-amine
(4aR,7aS)-1-(2-hydroxyethyl)-4-[3-(3-methoxyphenyl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(1,4-dithiepan-6-yl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
5-chloro-2-[4-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-2,3-dihydro-1H-indole
[(5-ethylpyridin-2-yl)methyl]({[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl})methylamine
3-{[2-(4-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}quinoline
2-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]pyrrolidin-2-yl}pyridine
2-[3-(1H-imidazol-1-yl)propyl]-9-[(2E)-3-phenylprop-2-en-1-yl]-2,9-diazaspiro[5.5]undecan-3-one
N3-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-1-cyclohexyl-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
methyl 1-{[4-(4-phenylbenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-4-carboxylate
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
3-{1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]piperidin-3-yl}benzoic acid
8-(4-fluoro-3-methylbenzoyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-[(1S,2S)-2-(benzyloxy)cyclohexyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-N-(4-methoxyphenyl)piperidin-3-amine
N-methyl-2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-(thian-4-yl)acetamide
N-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(1-ethylpiperidin-4-yl)acetamide
ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})[3-(methylsulfanyl)butyl]amine
methyl (2R)-2-[2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamido]propanoate
1-acetyl-N-{[1-(cyclopropylmethyl)piperidin-4-yl]methyl}piperidine-4-carboxamide
(1R,5S)-8-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}-3,8-diazabicyclo[3.2.1]octane
N-[(2R)-1-hydroxy-1,1-diphenylpropan-2-yl]imidazo[1,2-a]pyridine-6-carboxamide