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2-[2-(3-methylphenyl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-1,2-dimethylpiperazine
2-(9H-fluoren-2-ylmethyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
3-(diphenylmethyl)-5-(oxolane-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-methyl-5-(pyridin-4-yl)-N-(pyrimidin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
7-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
1-propanoyl-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}piperidine-3-carboxamide
N3-[(4-chlorophenyl)(phenyl)methyl]-1-cyclopentyl-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
methyl 3-{[2-(3-chlorophenyl)acetamido]methyl}-5-(furan-2-amido)benzoate
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-5-(hydroxymethyl)furan-2-carboxamide
N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-2H-1,3-benzodioxole-5-carboxamide
5-{[(2,5-difluorophenyl)methyl]amino}-1-methyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(2-methoxy-5-methylphenyl)-2-[4-(pyridin-4-yl)piperidin-1-yl]acetic acid
9-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-cyclopropyl-N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-5-oxopyrrolidine-3-carboxamide
N-({1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-3-yl}methyl)butanamide
3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]-4-(3-phenylpropyl)piperazin-2-one
2-methoxy-2-phenyl-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethan-1-one
2-methyl-5-({4-[4-(prop-2-en-1-yl)piperazine-1-carbonyl]-1,3-oxazol-2-yl}methoxy)-1,3-benzothiazole
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}quinoxaline-6-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylacetamide
ethyl (2S)-2-[2-(4-butanamidophenyl)acetamido]propanoate
methyl 3-[2-amino-3-cyano-6-(furan-2-yl)pyridin-4-yl]benzoate
1-(cyclopropylmethyl)-N-ethyl-5-{[3-(2-hydroxyethoxy)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]pyrrolidin-3-yl]methanol
3-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
4-(5-{[benzyl(methyl)amino]methyl}-1,2-oxazole-3-carbonyl)-3-ethyl-1-methylpiperazin-2-one
4-{5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperazine-1-carbaldehyde
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
3-{5-[(2,4,5-trimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
6-ethyl-3-[4-(furan-2-carbonyl)-1,4-diazepane-1-carbonyl]-1,5-dimethyl-1,2-dihydropyridin-2-one
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
methyl 1-[(3R,5S)-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[2-(1H-imidazol-1-yl)ethyl]amine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
5-{[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}-N-methylfuran-2-carboxamide
N-[(4,6-dimethylpyridin-2-yl)methyl]-4-(2,6-dimethylpyridin-3-yl)-N-methylpyrimidin-2-amine
5-ethyl-3-{[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
1-methyl-3-(propan-2-yl)-N-{2-[3-(trifluoromethyl)phenyl]ethyl}-1H-pyrazole-5-carboxamide
2-(4-hydroxypiperidin-1-yl)-6-(3-methylphenyl)-N-(2-phenylpropyl)pyridine-3-carboxamide
6-methyl-N-[1-(thiophene-2-carbonyl)piperidin-3-yl]imidazo[1,2-a]pyridine-2-carboxamide
1-(morpholin-4-yl)-3-[1-(2-phenylethyl)piperidin-3-yl]propan-1-one
1-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
(3R,4R)-N-[(2-aminopyrimidin-5-yl)methyl]-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-N,1-dimethylpyrrolidine-3-carboxamide
2-[(4-chlorophenyl)methyl]-N-(3-hydroxypropyl)-1,3-benzoxazole-5-carboxamide
3-hydroxy-1-(3-phenylpropyl)-3-[({pyrazolo[1,5-a]pyrimidin-3-ylmethyl}amino)methyl]piperidin-2-one
3-chloro-5-[2-(4-chlorophenyl)morpholine-4-carbonyl]-1,2-dihydropyridin-2-one
4-(1H-imidazol-2-yl)-1-[2-(1H-imidazol-2-yl)benzoyl]piperidine
2-(2H-1,3-benzodioxol-5-yloxy)-1-{3-[4-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one