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7-(cyclobutylmethyl)-2-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(dimethylamino)ethyl]-N-methyl-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
8-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
5-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxylic acid
3-[(1-methylpyrrolidin-3-yl)methyl]-1-(2-phenylphenyl)urea
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-(pentan-3-yl)pyridine-4-carboxamide
N-cyclooctyl-3-{[2-(1H-imidazol-4-yl)ethyl]amino}propanamide
4-cyclopropyl-6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
5-[(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-[(3-fluorophenyl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
2-[4-(4-carbamoylphenyl)-1H-pyrazol-1-yl]propanoic acid
methyl (2S,4S)-1-[(3-fluorophenyl)methyl]-4-(3-methoxybenzamido)pyrrolidine-2-carboxylate
4,4,4-trifluoro-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]butanamide
(3-{[1-(1H-indol-5-ylmethyl)pyrrolidin-3-yl]methyl}phenyl)methanol
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-2-(4-methylphenoxy)ethane-1-sulfonamide
methyl 3-({[4-(1H-imidazol-1-yl)phenyl]formamido}methyl)-5-(3-methoxybenzamido)benzoate
1-(3-chlorophenyl)-5-methyl-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-2-one
(1S,5R)-3-(pyridin-3-ylmethyl)-6-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
7-(3-methoxyphenyl)-2-[3-(pyrrolidin-1-yl)propyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-(5-methyl-4-{2-[3-(methylsulfanyl)phenyl]acetyl}-2-oxopiperazin-1-yl)benzonitrile
2-butyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,3-benzoxazole-5-carboxamide
3-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyridin-2-amine
4-hydroxy-N-(isoquinolin-5-ylmethyl)-N-methyl-2-(pyridin-2-yl)pyrimidine-5-carboxamide
(2S,3R)-2-[(2,6-dimethylquinolin-3-yl)formamido]-3-hydroxybutanoic acid
N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}-1H-1,2,3-triazole-5-carboxamide
1-(adamantan-1-yl)-4-[(1-ethyl-1H-imidazol-2-yl)methyl]piperazine
1-(3,6-dimethylpyrazin-2-yl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
1-[4-({2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl}methyl)phenyl]imidazolidin-2-one
N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(2H-1,2,3-benzotriazol-2-yl)-N-[(dimethyl-1,2-oxazol-4-yl)methyl]acetamide
N-{2-[7-(1-benzothiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}furan-3-carboxamide
3-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
1-ethyl-3-(propan-2-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-pyrazole-5-carboxamide
3-[1-(propan-2-yl)-1H-imidazol-2-yl]-1-[4-(propan-2-yl)benzoyl]piperidine
1-(5-methyl-1,3,4-oxadiazole-2-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidine
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-2-(pyrrolidin-3-yl)benzamide
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-phenylpiperazine
2-(4-chlorophenyl)-4-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}morpholine
(2S,3R)-2-amino-1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-hydroxybutan-1-one
1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-5-methoxyfuran-2-carboxamide
4-[4-(1H-pyrazol-3-yl)benzoyl]-1,4-oxazepan-6-ol
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(1H-1,2,4-triazol-3-ylmethyl)piperidine-3-carboxamide
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl]-6-ethyl-2-methylquinoline
6-methyl-2-(piperidin-1-yl)-N-[1-(pyridin-3-yl)propyl]pyrimidin-4-amine
methyl 6-(but-3-enoyl)-2-{[(3-chlorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-ethyl-6-[4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]pyrimidine
3-(1-benzyl-5-oxopyrrolidin-3-yl)-4-(4-ethylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one