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3-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-4-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(oxan-4-yl)piperidine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-(2-phenylethyl)-1,3-oxazole-4-carboxamide
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4,4,4-trifluorobutanamide
N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-(2-methylphenoxymethyl)piperidine-1-carboxamide
2-(3-{[4-(4-fluorophenyl)-1,4-diazepan-1-yl]methyl}phenoxy)ethan-1-ol
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(morpholin-2-yl)ethan-1-one
2-(dimethylamino)-2-(3-fluorophenyl)-1-(thiomorpholin-4-yl)ethan-1-one
[3-(2-methoxyethyl)-1-(pyridine-4-carbonyl)piperidin-3-yl]methanol
2-({8-methylimidazo[1,2-a]pyridin-2-yl}formamido)-N-(1,3-thiazol-2-yl)acetamide
8-(butan-2-yl)-1-(2-methoxyethyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-{4-[(dipropylamino)methyl]benzoyl}morpholin-2-yl)ethan-1-amine
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)urea
2-methoxy-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
(3S,5S)-1-[2-(propan-2-ylsulfanyl)acetyl]-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
1-cyclopentyl-4-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
3-[(1-ethyl-1H-indol-4-yl)methyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
N-(2H-1,3-benzodioxol-5-yl)-1-[(2,3,4-trimethoxyphenyl)methyl]piperidin-3-amine
1'-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
8-fluoro-2-{[2-(trifluoromethyl)morpholin-4-yl]methyl}-1,4-dihydroquinolin-4-one
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(1-benzothiophen-2-ylmethyl)-N-methyl-1-(2-methylpropyl)pyrrolidine-2-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(2-methanesulfonylethyl)pyrrolidin-3-yl]-3-methyl-1,2-oxazole-5-carboxamide
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-4-(piperidin-1-ylmethyl)benzamide
3-methyl-7-(2-methyl-2-phenoxypropanoyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-[(5-ethylpyridin-2-yl)methyl]-4-(4-fluoro-2-methylphenoxy)piperidine-4-carboxylic acid
(2R,6R)-11-methoxy-4-(morpholine-4-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-(1,2,3,6-tetrahydropyridine-1-carbonyl)pyrrolidine-2-carboxylic acid
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-(5-methyl-1H-pyrazol-1-yl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
2-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]pyridine-4-carboxamide
N,4,5-trimethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-(1H-pyrrol-1-yl)thiophene-3-carboxamide
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(1H-indol-3-yl)ethan-1-one
(4aS,7aR)-1-(1H-imidazol-2-ylmethyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopropyl-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
N3-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]piperidine-1,3-dicarboxamide
methyl[(3-{2-[4-(2-methyl-1,3-thiazole-4-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](naphthalen-1-ylmethyl)amine
(4aR,8aS)-1-[(3,4,5-trimethoxyphenyl)methyl]-6-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetamide
1-[2-(methylsulfanyl)ethyl]-4-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperazine
1-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pentan-1-one
1-cyclopentyl-4-{4-methoxy-2-[2-(methoxymethyl)piperidine-1-carbonyl]phenoxy}piperidine
1-(5-methylpyridin-3-yl)-3-[1-(pyrrolidin-1-ylmethyl)cyclohexyl]urea
5-{4-[4-(2-methoxyethyl)phenoxymethyl]phenyl}pyrimidin-2-amine
N-({1-[(2E)-3-(4-methoxyphenyl)prop-2-enoyl]piperidin-3-yl}methyl)furan-2-carboxamide
N-(3-carbamoylphenyl)-2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carboxamide
4-(furan-3-ylmethyl)-2-(2-phenylethyl)morpholine
2-chloro-5-{1-[(1-propylpiperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}pyridine
N-[(4-methylphenyl)(pyridin-4-yl)methyl]oxane-4-carboxamide