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3-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanoyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
5-methoxy-1-methyl-N-[1-(4-methylpyridin-2-yl)propyl]-1H-indole-2-carboxamide
1-[4-(4-chlorophenoxy)piperidin-1-yl]-4-(1H-imidazol-1-yl)butan-1-one
2-{4-[(2-methoxyphenyl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
1-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}-N-[(3R)-pyrrolidin-3-yl]piperidin-4-amine
5-(2-chlorophenyl)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]furan-2-carboxamide
4-[(1-methyl-1H-imidazol-5-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(4-fluorophenyl)methyl]pyrimidin-2-amine
1-(propan-2-yl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1H-pyrazole-4-carboxamide
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}piperidine-1-sulfonamide
N-{4-[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]-2-methylphenyl}pentanamide
5-methoxy-2-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4H-pyran-4-one
1-(4-{5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazin-1-yl)ethan-1-one
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1H-imidazol-2-ylmethyl)-N-methylacetamide
5-[2-(3-aminopyrrolidin-1-yl)pyrimidin-4-yl]-2-ethoxybenzoic acid
N-{[2-(4-acetylpiperazin-1-yl)-7-methoxyquinolin-3-yl]methyl}-2-ethyl-N-(2-methoxyethyl)butanamide
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1-phenyl-1H-pyrazole-4-carboxamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]methanol
1-(4-methylphenyl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperazin-2-one
1-[(4-methylphenyl)methyl]-4-[3-(pyridin-2-yl)propanoyl]piperazin-2-one
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
N-cyclopentyl-N-{[3,5-dimethoxy-4-(oxolan-2-ylmethoxy)phenyl]methyl}-4-(1H-pyrazol-1-yl)benzamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-amine
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-[4-(trifluoromethoxy)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(1H-1,3-benzodiazol-2-ylmethyl)-N-methyl-3-(piperidin-4-ylmethyl)benzamide
2-[5-(5-ethyl-1,2-oxazol-3-yl)-1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-3-yl]acetamide
N-(pyridin-3-yl)-2,3-dihydro-1,4-benzodioxine-6-carboxamide
N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2-(1-propylpiperidin-4-yl)acetamide
2-[3-(2-methylphenyl)-1H-pyrazol-1-yl]-N-(1-propyl-1H-indazol-3-yl)acetamide
2-(dimethylamino)-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-4-methylpyrimidine-5-carboxamide
9-(2-hydroxypyridine-3-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{8-fluoro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-3-methoxybenzamide
5-ethyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
(4aS,7aR)-1-(1,2-oxazole-3-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[4-(morpholin-4-yl)phenyl]methyl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
4-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-one
2-cyclobutyl-5-[3-(propoxymethyl)pyrrolidin-1-yl]-1,3,4-oxadiazole
2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)-1-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethan-1-one
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-(furan-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
3-[(3R,4S)-3-[(azepane-1-sulfonyl)amino]-4-cyclopropylpyrrolidin-1-yl]propanamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
5-[3-(methylsulfanyl)phenyl]-1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
2-ethyl-4-phenyl-9-(pyridazine-3-carbonyl)-2,9-diazaspiro[5.5]undecane
N4-[1-(3,4-dimethoxyphenyl)propyl]-5-methylpyrimidine-2,4-diamine
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3-(5-methyl-1H-pyrazol-1-yl)propanamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-3,4-dihydroquinazolin-4-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
7-[2-(thiophen-2-yl)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide