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4-(3-methyl-1,2,4-oxadiazol-5-yl)-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
2-amino-N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
6-({2-cyclopentyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-(3-methoxypropyl)-2-(3-methylpyridin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
4-benzyl-3-ethyl-1-[(2-ethylpyrimidin-5-yl)methyl]-1,4-diazepan-5-one
1-phenyl-2-({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethan-1-ol
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
(3R,4R)-4-cyclobutyl-3-methyl-1-(trimethylpyrimidin-4-yl)piperidin-4-ol
2-(4-acetylpiperazin-1-yl)-2-[3-(butylcarbamoyl)phenyl]acetic acid
1-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
N-(2-methoxyethyl)-2-methyl-3-({methyl[(5-methylthiophen-2-yl)methyl]carbamoyl}amino)benzamide
4-methoxy-N-(2-methoxyethyl)-2-{[1-(1-methoxypropan-2-yl)piperidin-4-yl]oxy}benzamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-[(3,4,5-trimethoxyphenyl)methyl]-1H-pyrazole-4-carboxamide
(3S,4R)-4-(2-methoxyphenyl)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]pyrrolidine-3-carboxylic acid
4-cyclobutyl-6-methyl-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]pyrimidin-2-amine
({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)(methyl)(quinolin-4-ylmethyl)amine
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]urea
4-(3-phenylphenyl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine
3-[1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-4-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
(3S,5R)-N3-(2H-1,3-benzodioxol-5-ylmethyl)-N5-(2,3-dihydro-1H-inden-5-yl)-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
N-cyclopropyl-N-[(5-methylthiophen-2-yl)methyl]-2-(1H-1,2,4-triazol-1-yl)acetamide
7-methoxy-3-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-2-(3-methylphenyl)quinoline
methyl 3-({4-[2-(4-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxy)ethyl]piperazin-1-yl}sulfonyl)thiophene-2-carboxylate
2-methyl-4-{4-[(2S)-2-(morpholine-4-carbonyl)pyrrolidine-1-carbonyl]phenyl}butan-2-ol
6-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}pyridine-3-carboxylic acid
4,6-dimethyl-2-{4-[2-methyl-2-(morpholin-4-yl)propyl]piperazin-1-yl}pyridine-3-carbonitrile
1-({5-[(2,6-difluoro-3-methylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-propylpiperidine
N-methyl-N-(3-methylbutyl)-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-ethyl-1-[3-(1H-pyrazol-1-yl)phenyl]urea
4-{2-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
2-(4-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-amido}-3,5-dimethyl-1H-pyrazol-1-yl)acetic acid
1-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-2,3-dihydro-1H-indol-2-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{1-[(2-methylphenyl)methyl]cyclopropyl}acetamide
3-{[ethyl(pyridin-2-ylmethyl)amino]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
(3R,4S)-4-(4-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1,4-diazepan-1-yl)oxolan-3-ol
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-3-ol
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]propan-1-one
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-{[6-(pyrrolidin-1-yl)pyridazin-3-yl]oxy}acetamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-7-methoxy-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
8-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1-oxa-8-azaspiro[4.6]undecane
1-{1-[(1,5-dimethyl-1H-indol-2-yl)methyl]piperidin-4-yl}piperidin-4-ol
1-butyl-4-(piperidin-4-ylmethyl)piperazin-2-one
2-(3-oxopiperazin-1-yl)-N-(quinolin-6-ylmethyl)acetamide
4-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propyl-1,4-dihydroquinoline-2-carboxamide
3-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-[2-(piperidin-1-ylmethyl)phenyl]urea
1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-2-(1-methylpiperidin-2-yl)ethan-1-one