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3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-2-oxopiperidin-1-yl]-2,2-dimethylpropanoic acid
6-methyl-2-[1-(2-methylfuran-3-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]{[3-(pyridin-2-ylmethoxy)phenyl]methyl}amine
1-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
N3-ethyl-N5-[(3-fluorophenyl)methyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]-1-cyclohexyl-3-(cyclopropylmethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
[(3R,4R)-1-[(2,3-difluorophenyl)methyl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
4-{2-amino-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1λ6-thiomorpholine-1,1-dione
4-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}thiomorpholine
(2S)-4-(methylsulfanyl)-2-({2-methylthieno[2,3-d]pyrimidin-4-yl}amino)butan-1-ol
5-({1-methyl-2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]pyrazolo[1,5-a]pyridine-7-carboxamide
5-(2-chlorophenyl)-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}furan-2-carboxamide
2-methyl-N-[2-(pyridin-4-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
2-[(4-chlorophenyl)methyl]-N-[2-(1H-pyrazol-4-yl)ethyl]-1,3-benzoxazole-5-carboxamide
4-(1H-imidazol-1-yl)-1-(pyrrolidine-1-sulfonyl)piperidine-4-carboxylic acid
2-methyl-N-[3-(2-propoxyphenyl)propyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-ethyl-1H-imidazol-1-yl)ethan-1-one
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-2,1-benzoxazole-3-carboxamide
5-cyclobutyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1,3,4-oxadiazol-2-amine
2-methyl-5-{2-[3-(1H-pyrazol-3-yl)phenyl]phenyl}-1,3,4-thiadiazole
1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
8-(3-hydroxy-4-methylbenzoyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{4-oxo-4-[3-(phenylamino)piperidin-1-yl]butyl}piperidin-2-one
methyl 5-[(3-hydroxy-3-methylbutan-2-yl)amino]-3-(4-methoxybenzamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(pyridin-4-yl)propanamide
N,2,2-trimethyl-N-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}oxan-4-amine
N-benzyl{[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]amino}sulfonamide
N-[(2-chlorophenyl)methyl]-3-{1-[3-(dimethylamino)benzoyl]piperidin-3-yl}propanamide
2-(5-{[2-(3-chloro-2,6-difluorophenyl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
1-{[4-(methylsulfanyl)phenyl]methyl}-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
5-[(2,4-dimethoxyphenyl)methyl]-3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
1-(2-methoxyethyl)-1-(1-methylpiperidin-4-yl)-3-(2,3,4-trifluorophenyl)urea
2-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]thiophen-3-amine
2-ethyl-9-[1-(4-fluorophenyl)cyclopropanecarbonyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenol
N-(2-methoxyethyl)-N-(thiophen-3-ylmethyl)oxane-2-carboxamide
2,6-dimethyl-8-[(thiophen-3-ylmethyl)amino]octan-2-ol
4-{[3-hydroxy-3-(piperidin-1-ylmethyl)pyrrolidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
(3aR,6aS)-5-[(5-bromothiophen-2-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2S)-2-amino-2-cyclohexyl-1-(4-{[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
3-{5-[(2-chloro-4-fluorophenyl)methyl]-1,2,4-oxadiazol-3-yl}pyridazine
N-benzyl-N-(2-hydroxyethyl)-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
5-(1,3-diphenyl-1H-pyrazole-5-carbonyl)-N-(3-methoxypropyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(morpholine-4-carbonyl)-N-[3-(1,3-oxazol-5-yl)phenyl]piperidine-1-carboxamide
{[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl}[2-(pyridin-3-yloxy)propyl]amine
(4aS,7aR)-1-[2-(2,4-difluorophenyl)acetyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 2-({3-[3-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}amino)acetate
6-ethoxy-3-[(4-ethyl-2-methyl-3-oxopiperazin-1-yl)methyl]-1,2-dihydroquinolin-2-one