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1-(cyclopropylmethyl)-4-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine
N-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
methyl (2S)-2-({6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidin-3-yl}formamido)propanoate
7-(cyclopropylmethyl)-2-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
(2R)-2-amino-1-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-3-phenylpropan-1-one
[(4aS,8aR)-6-[4-(propan-2-yl)benzenesulfonyl]-decahydro-1,6-naphthyridin-4a-yl]methanol
(2R)-2-[(3-{[(3-methylthiophen-2-yl)methyl]amino}phenyl)formamido]propanamide
1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-2-(methylsulfanyl)ethan-1-one
1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-methylpiperidin-3-ol
1-(1,2,3,4-tetrahydronaphthalen-2-yl)-4-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
8-fluoro-2-({[(4-methylpyridin-2-yl)methyl]amino}methyl)quinolin-4-ol
4-[1-(1-benzothiophen-5-ylmethyl)-1H-imidazol-2-yl]pyridine
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(3-methyl-1H-pyrazol-1-yl)acetamide
6-methoxy-3-{[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2-ethoxyethyl)acetamide
(1S,5R)-6-(cyclopropylmethyl)-3-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
2-({4-[3-(pyrrolidin-1-yl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
6-fluoro-2-{[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}quinolin-4-ol
4-(cyclohexylmethyl)-3-(2-oxo-2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)piperazin-2-one
2-methyl-N-(2-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)propanamide
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]acetamide
2-(pyridin-2-yl)-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-[(3S,4R)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]-N-[(4-methoxyphenyl)methyl]propanamide
(1R,5R)-6-[(2-tert-butyl-5-carbamoylfuran-3-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-[benzyl(methyl)amino]-3-[5-({[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
N-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-8-fluoroquinoline-2-carboxamide
2-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]propane-1,3-diol
1-[1-(1,3-oxazole-4-carbonyl)-4-phenylpiperidin-4-yl]ethan-1-one
4-[3-(3-chlorophenyl)pyrrolidine-1-carbonyl]-1H-pyrazole
4-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-1-phenylpiperazin-2-one
6-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}quinoxaline
1-{3-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-[2-({[2-(dimethylamino)ethyl](methyl)amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
(3R)-3,4,4-trimethyl-1-(pyrrolidine-1-sulfonyl)pyrrolidin-3-ol
N-[4-(azepan-1-yl)butyl]-2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]acetamide
1-{[3-(3-fluorophenyl)oxolan-3-yl]methyl}-4-(2-methylphenyl)piperazine
2-(3-hydroxypropyl)-9-(1-methyl-1H-pyrazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
6-[2-fluoro-6-(propan-2-yloxy)phenyl]-4-(4-methylpiperazin-1-yl)quinazoline
[(3S,5R)-1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-3-yl]methanol
N-{2-[ethyl(methyl)amino]-2-methylpropyl}-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
4-(3-methylphenoxy)-1-(thiophene-2-carbonyl)piperidine-4-carboxylic acid
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-(1H-1,2,4-triazol-3-yl)benzamide
1'-(2-amino-6-methoxypyrimidin-4-yl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
8-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
1-{2-methoxy-5-[(4-methoxypiperidin-1-yl)methyl]phenoxy}-3-(piperidin-1-yl)propan-2-ol
1-(1-benzoylpiperidin-4-yl)-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
1-(3-methylphenyl)-3-(2-phenylethyl)-N-(1,3,4-thiadiazol-2-yl)-1H-1,2,4-triazole-5-carboxamide
4-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1H-imidazole-2-carboxamide
5-(4-benzylpiperidin-1-yl)-1-methyl-N-[2-(morpholin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide