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1-(2-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{3-[3-(4-ethylpiperazin-1-yl)propyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}pyridine-3-carbonitrile
4-(2,3-dimethylphenyl)-5-ethyl-2-methylpyrimidine
N-[(5-methylpyrazin-2-yl)methyl]-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
4-[(furan-2-ylmethyl)amino]-5-methyl-N-[(1R)-1-phenylethyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-(3-ethoxypropyl)-5-methyl-4-[(pyridin-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
4-[5-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)-1,3-thiazol-2-yl]morpholine
methyl (1R,3S,3aR,6aS)-1,5-dimethyl-4,6-dioxo-3-(2-propoxyphenyl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-({7-[2-(4-chloro-2-methylphenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
2-[(2-fluorophenyl)methyl]-1,6-dimethyl-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
8-methoxy-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(2R)-1-(benzyloxy)-3-hydroxypropan-2-yl]-3-cyclopropaneamido-4-methylbenzamide
(cyclopropylmethyl)({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)amine
methyl (2S,4S)-1-methyl-4-(1-methyl-1H-indole-2-amido)pyrrolidine-2-carboxylate
3-methyl-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}furan-2-carboxamide
(5S,9aS,9bS)-2-[(4-methoxyphenyl)methyl]-5-(2-methyl-1,3-thiazol-5-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-methoxy-1-{4-[4-(pyridin-2-yl)pyrimidin-2-yl]-1,4-diazepan-1-yl}ethan-1-one
(1S,5R)-6-(2,5-dimethylfuran-3-carbonyl)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-{4-[2-(3-methoxypropyl)piperidine-1-carbonyl]phenyl}phenol
3-[1-(5-ethoxyfuran-2-carbonyl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 1-[(3R,5S)-5-{[2-(4-fluorophenyl)ethyl]carbamoyl}-1-(3-methylbut-2-en-1-yl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-[2-(4-fluorophenyl)-1-{1-[2-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}ethyl]-2-methoxy-N-methylacetamide
1-[1-(3-chlorobenzoyl)piperidin-4-yl]-N-cyclopropylpiperidine-4-carboxamide
4-({4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]furan-2-yl}methyl)morpholine
1-[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-3-(methoxymethyl)piperidine
1-(2-{3-[1-(1,4-dioxan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}phenyl)ethan-1-one
3,5-dimethyl-1-(1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}azetidin-3-yl)-1H-pyrazole
methyl 5-{[(3-fluorophenyl)methyl]carbamoyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-[2-({[3-hydroxy-2-oxo-1-(2-phenylethyl)piperidin-3-yl]methyl}amino)ethyl]acetamide
1-(2-methoxyethyl)-3-methyl-8-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
1-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
3-{1-[(2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
(2R,3S,6R)-3-phenyl-5-(1,3-thiazol-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl 3-(7-chloro-2-{[(1,5-dimethyl-1H-pyrazol-3-yl)formamido]methyl}-2,3-dihydro-1-benzofuran-5-yl)benzoate
2-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
9-[(5-methylthiophen-2-yl)methyl]-6-oxa-9-azaspiro[4.5]decane
1-(cyclopropylmethyl)-4-(2-ethoxypyridine-3-carbonyl)-2-(propan-2-yl)-1,4-diazepane
N-(1,3-benzoxazol-2-ylmethyl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
4-{3-[4-(4-chlorophenyl)-4-hydroxypiperidine-1-carbonyl]piperidin-1-yl}-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(isoquinolin-1-yl)piperidin-3-ol
methyl 5-{4-[3-(morpholin-4-yl)-3-oxopropyl]piperidin-1-yl}-5-oxopentanoate
4-{[5-(thiophene-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}thiomorpholine
6-methoxy-N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[4-(1-benzothiophen-3-yl)-2-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy]-N-(1,3-thiazol-2-ylmethyl)acetamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
4-{3-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]phenyl}phenol
methyl 4-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pentanoate
4-(1,3-dimethyl-4-{[3-(pyridine-2-carbonyl)piperidin-1-yl]methyl}-1H-pyrazol-5-yl)morpholine
5-methoxy-N,3-dimethyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-indole-2-carboxamide