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[4-(2,5-dimethyl-1-phenyl-1H-pyrrole-3-carbonyl)-1,4-oxazepan-6-yl]methanol
N-(oxolan-2-ylmethyl)-N-({4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)thiophene-2-carboxamide
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]butan-1-one
(4aS,8aR)-6-[2-(2-chlorophenoxy)acetyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
3-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]urea
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[1-(pyrazin-2-yl)propan-2-yl]acetamide
1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-4,4,4-trifluorobutan-1-one
2-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-[(3,5-dimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
2-amino-N-(2-methoxyethyl)-4-methyl-N-(thiophen-3-ylmethyl)-1,3-benzothiazole-6-carboxamide
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-methyl-8-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
8-[(2-chloro-6-fluorophenyl)methyl]-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(pyridin-4-yl)ethyl]amine
1-methyl-4-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperazine
4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-(pyridin-2-ylmethyl)benzamide
{4-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-1,4-oxazepan-6-yl}methanol
7-methoxy-3-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)quinolin-2-ol
1-{5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}-4-(pyridin-2-yl)piperidin-4-ol
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)[(3-phenyl-1H-pyrazol-4-yl)methyl]amine
1,5-dimethyl-4-{6-oxo-1-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
4-(2,3-dihydro-1H-inden-5-yloxy)-1-(6-methylpyridazin-3-yl)piperidine-4-carboxylic acid
methyl (2S,4S,5R)-5-(4-chlorophenyl)-1,2-dimethyl-4-(morpholine-4-carbonyl)pyrrolidine-2-carboxylate
2-[3-(1-benzofuran-2-yl)-4-methoxyphenyl]ethan-1-amine
{[2-(3-chlorophenyl)-6,7-dimethoxyquinolin-3-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
N-[1-(furan-2-ylmethyl)piperidin-4-yl]-2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
(2S,4S)-4-amino-N-methyl-1-(2-phenoxybenzoyl)pyrrolidine-2-carboxamide
2-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-3-yl]-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
4-methyl-N-[(3-methylphenyl)methyl]-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
3-(2H-1,3-benzodioxol-5-yl)-1-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]propan-1-one
3-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)-4-methoxyphenol
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
5-cyclobutanecarbonyl-1'-[(5-ethylpyridin-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
butyl(methyl){[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
4-[(2-methylprop-2-en-1-yl)oxy]-N-[2-(1H-1,2,4-triazol-1-yl)propyl]benzamide
{1-[4-(ethylamino)pyrimidin-2-yl]piperidin-4-yl}(pyridin-2-yl)methanol
7-(cyclopropylmethyl)-2-{2-methylthieno[3,2-d]pyrimidin-4-yl}-2,7-diazaspiro[4.5]decan-6-one
9-(1-benzofuran-5-ylmethyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
1,3-dimethyl-4-{2-oxa-7-azaspiro[4.5]decan-7-yl}-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid
1-(3-{[3-(5-chloro-2-methoxybenzoyl)piperidin-1-yl]methyl}phenyl)ethan-1-one
1-[(2-fluorophenyl)methyl]-5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
3-methyl-4-oxo-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-3,4-dihydroquinazoline-7-carboxamide
N-({1-[(2-methoxypyridin-3-yl)methyl]pyrrolidin-3-yl}methyl)pyridine-4-carboxamide
2-cyclohexyl-N-[3-(morpholin-4-yl)propyl]-1,3-benzoxazole-6-carboxamide
7-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-2-oxa-7-azaspiro[4.5]decane
8-chloro-2-({[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)quinolin-4-ol
2-(2-methyl-1,3-thiazol-4-yl)-1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]ethan-1-one
methyl 3-[(1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidin-4-yl)formamido]propanoate
2-(1H-pyrazol-1-ylmethyl)-4-(1H-1,2,3-triazole-5-carbonyl)-1,4-oxazepane
4-amino-2-{4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperazin-1-yl}pyrimidine-5-carbonitrile
3,5-dimethyl-4-(1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}pyrrolidin-2-yl)-1,2-oxazole