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3-ethyl-1-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)urea
N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}isoquinoline-1-carboxamide
1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
(2R)-2-phenyl-2-({5-propylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethan-1-ol
N-{2-methyl-5-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]phenyl}butanamide
7-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-2-oxa-7-azaspiro[4.5]decane
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N,2-dimethylpyridine-3-carboxamide
2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]acetamide
1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)urea
10-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
1-(2-methylfuran-3-carbonyl)-4-(pyridin-3-yl)piperidin-4-ol
4-{1-[(2,6-difluorophenyl)methyl]piperidin-4-yl}pyridine
N-[2-(3-phenylpropoxy)phenyl]pyridine-2-carboxamide
(3S)-3-{[5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]amino}azepan-2-one
3-(3-fluorophenyl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-2-(4-propanoylphenoxy)acetamide
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-4-ethenylbenzamide
ethyl 3-[(3-{3-oxo-3-[4-(pyridin-2-yl)piperazin-1-yl]propyl}piperidine-1-carbonyl)amino]propanoate
N-[(1R,3R)-3-aminocyclopentyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-(4-chlorophenyl)-N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]cyclopropane-1-carboxamide
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amine
2-(2H-1,2,3-benzotriazol-2-yl)-1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}ethan-1-one
3-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-1-[4-(thiophen-2-ylmethoxy)phenyl]urea
N-[(4,6-dimethylpyridin-2-yl)methyl]-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
N-(4-methylphenyl)-N'-[(4-methylphenyl)methyl]-N'-(prop-2-yn-1-yl)propanediamide
5-{[4-(1H-imidazol-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-fluoro-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}benzene-1-sulfonamide
3-methyl-6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-3H-imidazo[4,5-b]pyridine
3-[ethyl({[4-(6-oxo-4-propyl-1,6-dihydropyrimidin-2-yl)phenyl]methyl})amino]-1λ6-thiolane-1,1-dione
2-[({[(2-fluorophenyl)methyl]carbamoyl}amino)methyl]-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-{2-[4-(2-methoxyphenyl)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
5-ethyl-N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(thiophen-2-yl)propan-1-one
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(pyrazine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[(2-methyl-1,3-thiazol-4-yl)methyl]-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
1-[4-(thian-4-yl)piperazin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
5-(propan-2-yl)-N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
3-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-N-methyl-1,2,4-oxadiazole-5-carboxamide
(2S,3R)-2-amino-N-[1-benzyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-3-hydroxybutanamide
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}cyclobutanamine
1-(4-methylphenyl)-4-(5-methylthiophene-3-carbonyl)piperazin-2-one
1-(cyclobutylmethyl)-3-hydroxy-3-{[(1-phenylcyclopropyl)amino]methyl}piperidin-2-one
[(3R,4R)-1-(1-benzoxepine-4-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
(3S)-4-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3-dimethylpiperazin-2-one
2,3-dimethyl-N-(pyridin-3-yl)quinoxaline-6-carboxamide
1-(cyclohexylmethyl)-N-methyl-N-(quinoxalin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-(morpholin-4-yl)-6-[3-(propan-2-yloxy)phenyl]pyrimidin-2-amine
N-(oxan-4-yl)-4-(piperazine-1-carbonyl)benzene-1-sulfonamide
N-({2-[(dimethylamino)methyl]phenyl}methyl)-5,6-dimethylpyrimidin-4-amine