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1-{2-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-{4-[hydroxy(pyridin-3-yl)methyl]piperidin-1-yl}ethan-1-one
ethyl 1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-3-(3-phenylpropyl)piperidine-3-carboxylate
N-(1,3-dihydro-2-benzofuran-5-yl)-4-(oxolane-2-carbonyl)-1,4-diazepane-1-carboxamide
(2-methoxyethyl)({[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl})(thiophen-2-ylmethyl)amine
methyl 2-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane-7-carboxylate
(4aS,7aR)-1-(1H-indole-2-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[(5-methylthiophen-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[4-(4-benzylpiperidine-1-carbonyl)piperidin-1-yl]-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-{[(1R,2S,5R)-6,6-dimethylbicyclo[3.1.1]heptan-2-yl]methyl}-2-(methylamino)pyrimidine-5-carboxamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-(dimethylamino)pyridine-3-carboxamide
N-{[4-(dimethylamino)oxan-4-yl]methyl}-5-(oxolan-2-yl)thiophene-2-carboxamide
4-[5-(3-methoxyphenyl)furan-2-carbonyl]-1,4-oxazepan-6-ol
(1S,5R)-6-[(3-chloro-4,5-dimethoxyphenyl)methyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
8-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)imidazo[1,2-a]pyridine-2-carboxamide
(4aS,8aS)-2-[1-(3,4-difluorophenyl)piperidin-4-yl]-decahydro-2,7-naphthyridin-4a-ol
2-(2,5-dioxoimidazolidin-1-yl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]acetamide
N-ethyl-5-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrimidin-2-amine
1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]butan-2-ol
4-methoxy-3-{1H-pyrrolo[2,3-b]pyridin-4-yl}benzoic acid
2-{2-methyl-6-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]pyrimidin-4-yl}ethan-1-amine
methyl 3-{[(2-methyl-1,3-thiazol-4-yl)formamido]methyl}-5-[2-(1H-pyrazol-1-yl)acetamido]benzoate
N,1,3-trimethyl-N-[(3-methylpyridin-4-yl)methyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
{4-[(2-chlorophenyl)methyl]-1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl}methanol
2-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}benzoic acid
2-(dimethylamino)-N-methyl-2-(2-methylphenyl)-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
3-methyl-2-({4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
1-methyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-1H-pyrazole-4-carboxamide
1-methyl-4-{2-[4-(1H-pyrazol-5-yl)phenyl]pyridine-4-carbonyl}piperazine
6-(isoquinolin-5-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N-benzyl-N-methyl-3-({[2-(2-oxoimidazolidin-1-yl)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
4-{9-methoxy-7-oxo-3-[(2E)-3-phenylprop-2-en-1-yl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperazin-2-one
1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}-3-{[(pyridin-2-ylmethyl)amino]methyl}piperidin-2-one
2-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]ethan-1-ol
(1R,5S)-3-benzyl-6-[(2-methyl-1H-imidazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(4-methoxy-2-methylphenyl)methyl]-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine
3-[(4S)-2,5-dioxoimidazolidin-4-yl]-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]propanamide
(3S,4R)-1-[(4-acetylphenyl)methyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
2-{4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methylphenyl]phenyl}-2-hydroxyacetic acid
N-[(1S)-2-hydroxy-1-phenylethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
2-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}pyridine-3-carboxamide
1'-(4-methylquinolin-2-yl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
4-[(2-cyclohexylpyrimidin-5-yl)methyl]-1-methylpiperazine-2-carboxylic acid
2-(dimethyl-1,3-thiazol-5-yl)-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
5-{4-[1-(furan-2-ylmethyl)piperidin-4-yl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
4-fluoro-N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]benzene-1-sulfonamide
N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
4-(5-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2,4-oxadiazol-3-yl)pyridine
3-(4-chlorobenzoyl)-1-[(3,4,5-trimethoxyphenyl)methyl]piperidine