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2-(methylamino)-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-1,3-thiazole-4-carboxamide
N-methyl-N-{[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}cyclopentanamine
2-(6-methoxynaphthalen-2-yl)-4-(2-methoxypyridine-3-carbonyl)morpholine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}acetamide
1-(5-{5-methylthieno[2,3-d]pyrimidin-4-yl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl)pyrrolidine
1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-N-(oxan-4-ylmethyl)piperidine-4-carboxamide
6-methoxy-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}pyrimidin-4-amine
6-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine-2,4-diamine
N-[(2-ethoxypyridin-3-yl)methyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
1-methyl-6-oxo-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]-1,6-dihydropyridine-3-carboxamide
1-(2-aminopyridine-4-carbonyl)-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
4-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)-1-(4-methylphenyl)piperazin-2-one
{4-[4-(4-chlorophenoxy)piperidine-4-carbonyl]morpholin-3-yl}methanol
1-[5-benzyl-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,4-diazepan-5-one
(9aS)-2-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine
2-ethyl-9-[(4-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[4-(5-methylfuran-2-yl)benzoyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
(7R,9aR)-7-[(1S)-1-hydroxyethyl]-6,9-dioxo-N-phenyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
8-[2-(methylsulfanyl)acetyl]-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-2,6-dimethylpyridine-4-carboxamide
5-methyl-4-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1-propyl-1H-pyrazole
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(3,4-dimethoxyphenyl)ethan-1-one
5-(2-benzylmorpholine-4-carbonyl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
2-amino-6-(4-hydroxy-3-methoxyphenyl)-4-[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
1-ethyl-N-[2-(2-methoxyphenyl)ethyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
2-(2-chlorophenoxy)-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
5-methyl-3-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-3H,4H-thieno[2,3-d]pyrimidin-4-one
7-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-[(dimethylamino)methyl]-4-{1-[2-(pyrrolidin-1-yl)ethyl]-1H-imidazol-2-yl}phenol
methyl 4-{[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]carbamoyl}piperazine-1-carboxylate
1-{[5-(methoxymethyl)furan-2-yl]methyl}-3-(6-methoxynaphthalene-2-carbonyl)piperidine
4-(6-methoxypyridin-3-yl)-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
N-({8-[2-(2,5-dimethoxyphenyl)acetyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)pyridine-2-carboxamide
N-(1H-imidazol-2-ylmethyl)-5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
3-(2-ethyl-5-oxopyrrolidin-2-yl)-N-[1-(thiophen-2-yl)ethyl]propanamide
N-methyl-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-N-(pyridin-3-ylmethyl)propanamide
[(3R,4R)-1-[(4-chloro-2-fluorophenyl)methyl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
2-(ethoxymethyl)-N-[(2-ethoxypyridin-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-(5-ethylpyrimidin-2-yl)-2-(2-methoxyethyl)morpholine
[(5-chloro-2,4-dimethoxyphenyl)methyl][(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]methylamine
4-{2-[2-(1-benzofuran-2-yl)-1H-imidazol-1-yl]-1-(pyridin-4-yl)ethyl}morpholine
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-methanesulfonylpiperidine-4-carboxamide
2-(3-fluorophenoxy)-1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-6-oxopiperazine-2-carboxamide
2-(1-methylpyrrolidin-3-yl)-9-(thiophen-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(3-methoxyphenyl)amino]-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}butanamide
1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-4-(thiophen-2-yl)butan-1-one