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N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-(pyrazin-2-yl)propanamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-[2-(morpholin-4-yl)ethyl]acetamide
N-ethyl-3-(oxan-2-ylmethyl)benzamide
N-{2-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}acetamide
[(3-{2-[4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(naphthalen-1-ylmethyl)amine
6-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-9H-purine
8-acetyl-2-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(2R,3R,6R)-3-(4-fluorophenyl)-5-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
2-[(3R,4R)-3-hydroxy-4-(4-methylpiperazin-1-yl)piperidin-1-yl]pyridine-3-carboxylic acid
methyl 5-[4-ethyl-5-oxo-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]pentanoate
N-[3-(2-methylphenyl)phenyl]-4-(pyrrolidin-3-yl)piperazine-1-carboxamide
2-methyl-5-(2-{2-[(propan-2-yl)amino]ethyl}morpholin-4-yl)-2,3-dihydropyridazin-3-one
6,7-dimethoxy-N2-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)quinazoline-2,4-diamine
3-({1-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]pyrrolidin-3-yl}methyl)benzamide
2-methyl-9-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
(3aS,6aS)-2-[(2,4-dimethylphenyl)methyl]-5-(2-hydroxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(dimethylamino)-8-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-[4-(4-fluorophenoxy)piperidin-1-yl]-3-(1-methylpiperidin-3-yl)propan-1-one
N-[(2R,3R)-1'-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
N-(furan-2-ylmethyl)-5-methyl-N-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide
2-cyclobutyl-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-(pyridin-2-yl)-1-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}propan-1-one
(1S,5R)-N-[(4-methylphenyl)methyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]but-3-enamide
2-(ethylamino)-N,4-dimethyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-thiazole-5-carboxamide
N,6-dimethyl-2-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
9-[(2,4,6-trimethoxyphenyl)methyl]-1,4,9-triazaspiro[5.5]undecan-5-one
4-acetamido-N-[2-(4-ethylmorpholin-2-yl)ethyl]-2-methylbenzamide
4-(4-ethyl-1H-pyrazol-5-yl)-1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
2-[4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]ethan-1-ol
2-(2,5-dimethylphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
1-(furan-2-carbonyl)-4-[4-(pyridin-4-yl)pyrimidin-2-yl]-1,4-diazepane
4-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
1-(cyclopropylmethyl)-5-(2-methylphenyl)-1H,4H-pyrazolo[3,4-d]imidazole
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-ethylacetamide
N,N-dimethyl-4-{4-[(pyridin-2-ylmethyl)carbamoyl]phenoxy}piperidine-1-carboxamide
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-(1H-pyrazol-1-yl)propan-1-one
2-(dimethyl-1,2-oxazol-4-yl)-1-{3-[3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxymethyl]piperidin-1-yl}ethan-1-one
N-[3-(2-ethylphenoxy)propyl]-N,2,4-trimethylpyrimidine-5-carboxamide
N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}cyclohexanecarboxamide
(8R,9aS)-8-hydroxy-2-[2-(pyridin-2-yl)ethyl]-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
4-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-1-(4-methoxyphenyl)piperazin-2-one
3-{1-[1-(4-chlorophenyl)cyclobutanecarbonyl]piperidin-3-yl}-N-cyclopropylpropanamide
N-(4-fluoro-2-methylphenyl)-3-{1-[2-(pyridin-2-yl)acetyl]piperidin-3-yl}propanamide
2-{[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
1-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}morpholine-3-carboxamide
N-[(2-fluorophenyl)methyl]-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(4-methyl-1,3-thiazol-5-yl)-N-[1-(thian-4-yl)piperidin-4-yl]propanamide