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6-[4-(2-methoxyphenoxy)piperidin-1-yl]pyrimidine-2,4-diamine
dimethyl(2-{4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]morpholin-2-yl}ethyl)amine
2-{methyl[(1-methyl-1H-imidazol-2-yl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-[3-(difluoromethoxy)benzoyl]-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
3-methanesulfonyl-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
2-{1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidin-2-yl}-1,3-benzothiazole
2-{1-ethyl-5-[3-(1H-1,2,3,4-tetrazol-1-yl)phenoxymethyl]-1H-1,2,4-triazol-3-yl}acetamide
N-cyclobutyl-3-{[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]sulfamoyl}benzamide
2,5-dimethyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-{1-[6-(benzylamino)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
7-[(2,3-difluorophenyl)methyl]-2-(pyridine-2-carbonyl)-2,7-diazaspiro[4.5]decane
4-[(dipropylamino)methyl]-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}benzamide
(1S,5R)-6-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-(2-chloro-6-methoxyphenyl)pyrazolo[1,5-a]pyrimidine
4-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}benzoic acid
N-methyl-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2,1,3-benzothiadiazol-5-ylmethyl)({[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl})methylamine
2-(2-chlorophenyl)-5-methyl-4-{1H-pyrazolo[3,4-b]pyridin-1-ylmethyl}-1,3-oxazole
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-({methyl[2-(pyrrolidin-1-yl)ethyl]amino}methyl)piperidin-2-one
N-({3-[2-(dimethylamino)ethoxy]phenyl}methyl)-4-methyl-N-(pyridin-2-ylmethyl)-1,2,5-oxadiazole-3-carboxamide
2-{3-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidine-1-carbonyl]-5-methyl-1H-pyrazol-1-yl}-N-methylacetamide
(2R,6S)-4-[6-chloro-3-(pyrrolidin-1-ylmethyl)imidazo[1,2-a]pyridine-2-carbonyl]-2,6-dimethylmorpholine
N-(isoquinolin-5-ylmethyl)-2-(4-methoxyphenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
5-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-3-(5-methylthiophen-2-yl)-1H-pyrazole
4-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-5-ethyl-2-methylpyrimidine
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-3-(1H-pyrazol-1-yl)butan-1-one
5-(3,4-difluorophenoxymethyl)-N-(1H-imidazol-2-ylmethyl)-1,2-oxazole-3-carboxamide
4-{[methyl(oxolan-2-ylmethyl)amino]methyl}-N-(1-methyl-1H-pyrazol-4-yl)benzamide
4-(2-{1-[(2-ethylpyrimidin-5-yl)methyl]piperidin-2-yl}ethyl)phenol
(2S)-2-[(8-fluoroquinolin-2-yl)formamido]-3-(4-hydroxyphenyl)propanamide
[1-(1-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidin-3-yl)piperidin-4-yl]methanol
5-[(4-benzylpiperidin-1-yl)methyl]-N-cyclopropyl-1,2-oxazole-3-carboxamide
2-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(2-oxopiperidin-1-yl)acetamide
1-cyclopentyl-N-[(1-ethyl-1H-indazol-3-yl)methyl]-6-oxopiperidine-3-carboxamide
2-tert-butyl-4-hydroxy-N-(isoquinolin-5-ylmethyl)-N-methylpyrimidine-5-carboxamide
1-ethyl-4-({2-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-1,4-diazepane
methyl 1-{3-[(2,4-difluorophenyl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
N-[1-({5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)piperidin-4-yl]pyridin-2-amine
N-({3-[(2-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)-1-methyl-4-oxo-N-(pyridin-4-ylmethyl)-1,4-dihydroquinoline-3-carboxamide
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-propoxyethan-1-one
1-(2,3-dichlorobenzoyl)-4-(1-ethyl-1H-imidazol-2-yl)piperidine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
2-{2-[(dipropylamino)methyl]phenyl}-6-ethyl-3,4-dihydropyrimidin-4-one
1-[(4aR,8aS)-1-[2-(thiophen-3-yl)acetyl]-decahydro-1,6-naphthyridin-6-yl]-4-phenylbutan-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,3,5,7-tetramethyl-1H-indole-2-carboxamide
methyl 1-(naphthalen-2-ylmethoxy)-2-oxo-8-(1,3-thiazol-2-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
7-(1H-inden-2-yl)-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[4-(propylsulfanyl)phenyl]-4-(pyridin-3-ylmethoxy)piperidine-1-carboxamide
3-(4-methoxy-3,5-dimethylbenzoyl)-1-propylpiperidine