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N-butyl-N-methyl-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
methyl (2S,4S)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(2-methylphenyl)methyl]pyrrolidine-2-carboxylate
[9-(1-methyl-1H-1,3-benzodiazole-2-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[(1,2-oxazol-3-ylmethyl)amino]pyridine-3-carboxamide
2-[2-(propan-2-yl)-1H-1,3-benzodiazol-1-yl]-N-[1-(pyrimidin-2-yl)piperidin-3-yl]acetamide
3-{[1-(pyridin-2-yl)piperidin-3-yl]methyl}-1-[4-(1H-1,2,4-triazol-1-yl)phenyl]urea
5-{4-[(dimethylamino)methyl]phenyl}-2-fluorobenzoic acid
4-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-1-phenylpiperazin-2-one
N-[4-(4-{[2-(1H-imidazol-1-yl)ethyl]amino}piperidin-1-yl)phenyl]-2-(4-methoxyphenyl)acetamide
N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-3-(2,5-dioxoimidazolidin-4-yl)propanamide
2-{4-[(2-fluorophenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
2-(dimethylamino)-4-methyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]pyrimidine-5-carboxamide
(1R,5R)-6-(2-methoxyethyl)-N-[2-(thiophen-2-yl)ethyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(4-chlorophenoxy)pyridine-3-carboxamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
1-(5-fluoro-2-methoxybenzoyl)-2-(3-methoxypropyl)piperidine
1-[1-(3-fluoropropyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-2-methyl-3-(1H-1,2,4-triazol-1-yl)propanamide
methyl 3-({1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}carbamoyl)benzoate
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamide
5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
{4-[2-chloro-5-(piperidin-1-yl)benzoyl]-1,4-oxazepan-6-yl}methanol
2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]-N-(quinolin-3-ylmethyl)acetamide
4-(2-oxopyrrolidin-1-yl)-N-(quinolin-8-yl)benzamide
1-[2-oxo-2-(3-phenylpiperazin-1-yl)ethyl]pyrrolidin-2-one
3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-N-cyclopropylpropanamide
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]ethan-1-one
N-[(3R,4S)-1-(2-methoxyethyl)-4-propylpyrrolidin-3-yl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
6-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]pyrazine-2-carboxamide
(3S,4S)-1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine-3,4-diol
9-(isoquinolin-1-yl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
3-(3,3-diphenylpiperidine-1-carbonyl)pyridine
4-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(3aS,6aR)-3-cyclopentyl-5-(thiophen-3-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-6-methyl-2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1,3-dimethyl-6-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
dimethyl({[(3S,4R)-1-(6-methylpyridine-2-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl})amine
1-[1-(2-cyanobenzoyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
2-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-6-fluorobenzamide
1'-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(2H-1,3-benzodioxole-5-carbonyl)-3-(3-fluoro-4-phenylbenzoyl)piperidine
8-[4-(pyrrolidin-1-yl)benzoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
benzyl 7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxylate
3-(2,5-dioxoimidazolidin-4-yl)-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]propanamide
2-(2H-1,3-benzodioxol-5-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
2-({3-amino-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-5-yl}methyl)-5-(dimethylamino)-2,3-dihydropyridazin-3-one
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N,N-diethylbenzamide