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1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]-3-(4-methoxyphenyl)propan-1-one
1-(4-aminoazepan-1-yl)-2-(naphthalen-1-yl)ethan-1-one
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-(1,2,4-oxadiazol-3-yl)piperidine
(3R,5S)-5-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]pyrrolidin-3-ol
6-{6,8-dioxo-2,7-diazaspiro[4.4]nonan-2-yl}pyridine-2-carbonitrile
3-[2-(piperidin-2-yl)ethyl]-5-[6-(pyrrolidin-1-yl)pyridazin-3-yl]phenol
1-{5-[5-(3-ethyl-1,2-oxazol-5-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}ethan-1-one
1-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}-2-(morpholin-2-yl)ethan-1-one
6-[1-(2,7-dimethylquinoline-4-carbonyl)piperidin-4-yl]-2-methyl-3,4-dihydropyrimidin-4-one
methyl 3-(cyclobutylmethoxy)-5-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]carbamoyl}benzoate
1-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]pentane-1,2-dione
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-[4-(trifluoromethyl)pyridin-2-yl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-3,3-dimethylbutanamide
4-{[3-(4-fluorophenoxymethyl)piperidin-1-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-methoxyacetamide
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)benzamide
1-{3-[2-(morpholin-4-ylmethyl)phenyl]phenyl}ethan-1-one
N,N-dimethyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
N-cyclopropyl-1-(2-{1-[2-(2-methylphenyl)acetyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
N-(2-methoxyethyl)-N-methyl-2-(1H-pyrazol-1-yl)benzamide
N-(2-chlorophenyl)-3-{[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}propanamide
N-cyclopropyl-1-[1-(1H-pyrazole-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
3-methoxy-1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
1-(3-{1-[2-(6-hydroxypyrimidin-4-yl)ethyl]-1H-imidazol-2-yl}-2,4,6-trimethylphenyl)ethan-1-one
2-methyl-5-{4-[4-(morpholin-4-yl)benzoyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
2-amino-5-methyl-6-(propan-2-yl)-4-(pyridin-4-yl)pyridine-3-carbonitrile
2-[2-(2-methyl-2,3-dihydro-1H-indol-1-yl)-2-oxoethyl]-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
(1S,5R)-6-(2-methoxyethyl)-3-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 2-{[5-acetamido-2-ethyl-1-(pyridin-3-ylmethyl)-1H-1,3-benzodiazol-7-yl]formamido}-4-(methylsulfanyl)butanoate
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[5-(4-methylphenoxymethyl)-1,3,4-thiadiazol-2-yl]urea
6-[3-(2-fluorophenyl)benzoyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
N-(1-benzylpyrrolidin-3-yl)-N,2,6-trimethylpyrimidine-4-carboxamide
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]pyrrolidin-3-yl]methanol
(3aS,6aS)-2-cyclopentanecarbonyl-5-[3-(methylsulfanyl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
ethyl 1-(cyclopropylmethyl)-5-[3-(2-methoxyphenyl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-(2-methoxyphenyl)-2-methyl-5-[3-(1H-pyrazol-4-yl)propyl]-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-1-{thieno[3,2-d]pyrimidin-4-yl}piperidine
3-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetamido]-N-(3-methoxyphenyl)benzamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-hydroxy-2-methylpropan-2-yl)acetamide
(3S,4R)-1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
1-[1-(methoxymethyl)cyclobutanecarbonyl]imidazolidin-4-one
3-(cyclopropylmethyl)-1-(2-methyl-5-sulfamoylbenzoyl)piperidine-3-carboxylic acid
6-{1-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]piperidin-4-yl}-2-methylpyrimidin-4-ol
(3S,4S)-1-{2-[1-(propan-2-yl)piperidin-4-yl]acetyl}-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
N-[2-(1-hydroxycyclopentyl)ethyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(1R,3S)-N3-ethyl-N1-(furan-3-ylmethyl)-1,2,2-trimethylcyclopentane-1,3-dicarboxamide
N-(5-{[4-(cyclohexylmethyl)-5-oxo-1,4-diazepan-1-yl]methyl}thiophen-2-yl)acetamide
N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(thiophene-2-sulfonamido)acetamide
2-[2-chloro-4-({4-[(methylcarbamoyl)methyl]piperidin-1-yl}methyl)phenoxy]propanoic acid