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1-{5-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]-2-methoxyphenoxy}-3-(piperidin-1-yl)propan-2-ol
2-(2,5-dimethylphenyl)-N-{[1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]methyl}acetamide
N3-benzyl-N3-(1,3-thiazol-2-ylmethyl)piperidine-1,3-dicarboxamide
4-[(2,6-dichlorophenyl)methyl]-1,4-oxazepan-5-one
N-(cyclohex-1-en-1-ylmethyl)-1-ethyl-5-oxopyrrolidine-3-carboxamide
4-{[3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]methyl}benzonitrile
N-cyclopropyl-1-(2-{1-[3-(dimethylamino)benzoyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
N,5,6-trimethyl-N-[1-(pyridin-3-yl)pentyl]pyridine-3-carboxamide
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
ethyl 4-[(4-{[1-(1-methyl-4-oxo-1,4-dihydroquinoline-3-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine-1-carboxylate
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,5-dimethyl-1,2-oxazole-4-carboxamide
2-(4-fluoro-2-methylphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
1-{7-[cyclohexyl(hydroxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(2H-indazol-2-yl)ethan-1-one
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(2,4-difluorophenyl)methyl]amino}-1-(2-methylpropyl)pyrrolidine-2-carboxamide
1-{[(5-acetyl-2-ethoxyphenyl)carbamoyl]amino}cyclopentane-1-carboxamide
6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxylic acid
1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
4-(4-{[3-(hydroxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}acetamide
2-{[5-(1-ethyl-1H-pyrazol-3-yl)-4-phenyl-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-(2,4-dimethoxyphenyl)propanamide
4-({1-[(furan-3-ylmethyl)(methyl)amino]hex-5-en-2-yl}oxy)-2-methoxypyridine-3-carbonitrile
8-[(3-fluoro-4-methoxyphenyl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-4-(thiophen-2-yl)butan-1-one
5-methyl-4-(4-methylpiperazin-1-yl)-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-1,3-thiazole-4-carboxamide
6-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-N,N-dimethylpyrazine-2-carboxamide
3-[(5-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}furan-2-yl)sulfanyl]-4-methyl-4H-1,2,4-triazole
3-[1-(2-chloropyridine-4-carbonyl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
5-methyl-N-(3-methylbutyl)-4-[(thiophen-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
3-(4-chloro-1H-pyrazol-1-yl)-1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]propan-1-one
2-{4-[(8-methylquinolin-5-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
3-methyl-5-{1-[2-(2-methyl-1-benzothiophen-3-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazole
9-{2-[ethyl(methyl)amino]acetyl}-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
[(3aS,6aS)-2-{2-methylthieno[3,2-d]pyrimidin-4-yl}-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
6-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidin-4-amine
4-ethyl-3-{1-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1,4-dioxan-2-ylmethyl)-5-[1-(2-ethylbutyl)-4-hydroxypiperidin-4-yl]-1-benzofuran-2-carboxamide
N-(1-benzylpyrrolidin-3-yl)-3-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)propanamide
(1S,2R)-1-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-2,3-dihydro-1H-inden-2-ol
3-hydroxy-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)propanamide
7-chloro-4-(8-fluoroquinoline-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl 4-[({1-[(3-fluorophenyl)methyl]-6-oxopiperidin-3-yl}formamido)methyl]benzoate
1-[cyclohexyl(methyl)amino]-3-[3-({[(2-fluorophenyl)methyl]amino}methyl)phenoxy]propan-2-ol
N-(1-hydroxybutan-2-yl)-6-methyl-N-[(5-methylthiophen-2-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
4-{2-[1-(thiophene-2-sulfonyl)piperidin-2-yl]ethyl}morpholine
1-[2-methoxy-6-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
2-amino-4-(2,3,4-trimethoxyphenyl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile