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2-ethyl-4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]pyridine
methyl 8-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2-({2-[1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
5-ethyl-2,3-dimethyl-N-[2-(pyrrolidin-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-[4-(oxolan-2-ylmethoxy)phenyl]urea
3-[(3S,4R)-4-(dimethylamino)-1-(2,2-diphenylethyl)piperidin-3-yl]-1-[4-(3-methoxyphenyl)piperazin-1-yl]propan-1-one
N,5-dimethyl-N-(oxolan-3-yl)-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
2-(4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazin-1-yl)-1,3-benzoxazole
1-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-2-(pyridin-4-ylsulfanyl)ethan-1-one
1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
5-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-5-oxopentanamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-5-(1H-indol-3-ylmethyl)-1-(2-methoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1S,4S)-2-(2-methoxy-5-methylphenyl)-5-[2-(naphthalen-1-yl)acetyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-ethyl-2,7-dimethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}pyrazolo[1,5-a]pyrimidine-5-carboxamide
N-(2-methoxyethyl)-2-(pyridine-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-[3-({[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)propyl]pyrrolidin-2-one
N6-benzyl-N5-methyl-N5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N,2-dimethyl-N-[1-(pyridin-3-yl)pentyl]-1,3-benzoxazole-6-carboxamide
N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
3-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
3-[2-(2-phenylethyl)pyrrolidine-1-carbonyl]-5-propyl-1,2-oxazole
(3R,4R)-N-[(4-fluorophenyl)methyl]-3-hydroxy-3,4-dimethylpyrrolidine-1-carboxamide
N-methyl-5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyridin-2-amine
2-phenyl-5-(4H-1,2,4-triazol-4-ylmethyl)-1,3,4-oxadiazole
5-oxo-1-phenyl-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,5-dihydro-1H-pyrazole-3-carboxamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(azocan-1-yl)acetamide
4-{5-[(carbamoylamino)methyl]-1-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl}benzamide
3-[({[1-(hydroxymethyl)cyclopropyl]methyl}(methyl)amino)methyl]-6,7-dimethoxy-1,2-dihydroquinolin-2-one
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperazine
N-{[6-chloro-4-(cyclopentylamino)quinazolin-2-yl]methyl}-2-(1H-imidazol-2-yl)benzamide
5-[(2S)-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl]-N,N-dimethylpyridin-2-amine
1-[3-(3-hydroxy-3-methylbutyl)benzoyl]azepan-4-ol
3-{2-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-[3-(3-methylphenyl)phenyl]-1-(oxan-4-yl)piperidine-3-carboxamide
3-[1-(carbamoylcarbonyl)piperidin-3-yl]-N-[(2,4-dimethoxyphenyl)methyl]propanamide
methyl 3-(oxolane-2-amido)-6-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
1-(cyclohexylmethyl)-N5-[2-(3-methoxyphenyl)ethyl]-N3,N3-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
[(5-chloro-2-methoxyphenyl)methyl](ethyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
4-(2-hydroxypropyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-amino-5-ethyl-4-(2-methoxypyrimidin-5-yl)-6-(propan-2-yl)pyridine-3-carbonitrile
(4aS,7aR)-1-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-(2-methoxyphenyl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)acetamide
N-(1-{7-[(2,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
3-[2-chloro-5-(pyrrolidine-1-carbonyl)phenyl]-1-methyl-1-(thian-4-yl)urea
2-[2-({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
7-(7-chloroquinolin-4-yl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-(4-ethylpiperazin-1-yl)acetamide
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-(1-carbamoylcyclopentyl)-3-(4H-1,2,4-triazol-4-yl)benzamide