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N-benzyl-1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-amine
(1S,4S)-2-(3-chloro-4-methoxyphenyl)-5-[2-(3-methoxyphenyl)acetyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-ethyl-3-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]propanamide
9-(azepane-4-carbonyl)-2-cyclobutyl-2,9-diazaspiro[5.5]undecan-3-one
N-{[(3S,4S)-3-hydroxy-1-[(3-methylthiophen-2-yl)methyl]piperidin-4-yl]methyl}-2,5-dimethylfuran-3-carboxamide
N-(3-chloro-4-methoxyphenyl)-3-[1-(pyrimidin-2-ylmethyl)piperidin-3-yl]propanamide
2-(azepan-1-yl)-1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-3,5-dimethoxy-N-(oxolan-2-ylmethyl)benzamide
7-[1-benzyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
(1S,5R)-6-(2-methoxypyridine-4-carbonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-3-(2-methylphenyl)propanamide
3-(azepane-1-carbonyl)-N-[(5-chlorothiophen-2-yl)methyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl)benzoic acid
(2S,4S)-4-amino-1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[(3-methoxyphenyl)methyl]-8-(thiophen-3-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
1-{1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-4-phenylpiperidin-4-yl}ethan-1-one
N-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3R,4R)-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-(phenylamino)pyrimidine-5-carboxamide
2,6-dimethyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}quinoline-4-carboxamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
2-[(1R,3S,3aS,6aR)-3-(5-tert-butyl-1H-pyrazol-3-yl)-1-(hydroxymethyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]ethan-1-ol
2-[4-(2-aminopyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)acetamide
1-{[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]methyl}-3-ethylurea
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-methoxypropanamide
2-(4-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1-cyclopentylpiperazin-2-yl)ethan-1-ol
1-(cyclohexylmethyl)-N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-6-oxopiperidine-3-carboxamide
[2-methyl-1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
7-{2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(5-methylfuran-2-yl)ethyl]benzamide
5-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
2-phenyl-N-(1-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
5-chloro-4-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-2-methylpyrimidine
(4aS,8aR)-6-{5-amino-[1,2,4]triazolo[4,3-c]pyrimidin-7-yl}-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
(2R,3R,6R)-5-benzoyl-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[2-(1-cycloheptanecarbonylpiperidin-3-yl)-1H-imidazol-1-yl]acetamide
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridin-3-ol
1-(2-oxo-2-{6-oxo-1H,2H,3H,4H,6H,10bH-pyrimido[2,1-a]isoindol-1-yl}ethyl)-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
8-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
1,3-dimethyl-N-[1-(3,4,5-trimethoxyphenyl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-(4-tert-butylbenzoyl)-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidine
N-(2-fluorophenyl)-3-(1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-3-yl)propanamide
2-ethyl-N-[2-(2-methylphenyl)-2-(4-methylpiperidin-1-yl)ethyl]pyrimidine-5-carboxamide
3-[2-(2-hydroxyethoxy)ethyl]-3,4-dihydroquinazolin-4-one
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-3-(pyridin-4-yl)propanamide
N-[(3S,4R)-3-benzyl-1-methylpiperidin-4-yl]-2-(1-ethylpiperidin-4-yl)acetamide
2-[1-(2H-1,3-benzodioxol-5-yl)-1H-imidazol-2-yl]-5-ethylpyridine
5-benzyl-5-[1-(furan-2-carbonyl)piperidin-4-yl]-3-[2-(pyrrolidin-1-yl)ethyl]imidazolidine-2,4-dione