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5-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidine-1-carbonyl}-N-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
3-methoxy-4-{2-[2-(pyridin-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}benzoic acid
2-[4-(5-acetylpyridin-2-yl)-1H-pyrazol-1-yl]-N-(1,3-dimethyl-1H-pyrazol-5-yl)acetamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
5-{3-[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]-3-oxopropyl}-5-(furan-2-ylmethyl)pyrrolidin-2-one
1-(2,3-dimethylquinoxalin-6-yl)-3-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}urea
2-{4-[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]piperidin-1-yl}acetic acid
1-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(cyclohex-1-en-1-yl)ethan-1-one
N-benzyl-1-(1-benzylpiperidin-4-yl)piperidine-3-carboxamide
(1R,9aR)-1-{[4-(3-methoxyphenyl)piperazin-1-yl]methyl}-octahydro-1H-quinolizin-1-ol
N-(1-benzyl-1H-pyrazol-3-yl)-2-[4-(1-methyl-1H-pyrazol-4-yl)-1H-pyrazol-1-yl]acetamide
4-[2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)acetyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)quinoline-8-sulfonamide
3-(2-methoxyethyl)-1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidine
1-ethyl-N-(furan-3-ylmethyl)-5-[(3-hydroxy-2,2-dimethylpropyl)amino]-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(azocan-1-yl)-3-(2H-1,3-benzodioxol-5-yl)-3-phenylpropan-1-one
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
methyl 6-{2-azabicyclo[2.2.1]heptan-2-ylmethyl}-3-(1,3-dimethyl-1H-pyrazole-5-amido)thieno[2,3-b]pyridine-2-carboxylate
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(1,2-oxazinan-2-yl)propanamide
ethyl[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl](methyl)({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
2-[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]-2-(dimethyl-1,2-oxazol-4-yl)acetic acid
N,2-dimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1-benzofuran-5-carboxamide
6-(4-ethylpiperazin-1-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
4-(2-fluorophenoxy)-1-{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}piperidine
3-bromo-5-(morpholine-4-sulfonyl)benzoic acid
(1H-1,3-benzodiazol-2-ylmethyl)(methyl){[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
(2R,3R)-1'-(1,2-oxazole-3-carbonyl)-3-(thiomorpholin-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-(2,3-dihydro-1H-inden-2-yl)-5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyethyl)-1H-1,2,4-triazole
(1R,5R)-3-cyclobutanecarbonyl-6-(furan-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole
6-methyl-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxylic acid
N,N-dimethyl-1-(2-methylpropyl)-5-{[3-(propan-2-yloxy)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(1R,3S)-3-ethoxy-7-(pyridine-4-carbonyl)-7-azaspiro[3.5]nonan-1-ol
N,2-dimethyl-6-(piperidin-4-yl)-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-4-amine
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine
2-(3-fluorophenoxy)-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]ethan-1-one
1-{4-[4-(2-ethyl-6-methylpyrimidin-4-yl)piperazin-1-yl]piperidin-1-yl}-2-methylpropan-1-one
N-(1-methanesulfonylpiperidin-4-yl)-8-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-methyl-4-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]benzene-1-sulfonamide
1-(2-methoxyphenyl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
3-(3,3-diphenylpiperidin-1-yl)propanamide
3-(1H-1,3-benzodiazol-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]propanamide
N-methyl-1-propyl-N-(1,3-thiazol-4-ylmethyl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazole
8-methanesulfonyl-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-amino-4-(2,3-dimethoxyphenyl)-6-(propan-2-yl)pyridine-3-carbonitrile
N-[2-(2-fluorophenyl)ethyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-(azocane-1-carbonyl)-N-phenylpyrimidin-2-amine
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]pyridin-2-amine