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methyl 1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-5-[(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
methyl 1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-phenylpyrrolidine-3-carboxylate
1-methyl-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-6-oxo-1,6-dihydropyridazine-3-carboxamide
2-[(3,4-difluorophenyl)methyl]-8-(oxan-4-yl)-2,8-diazaspiro[4.5]decan-3-one
1-methyl-3-[3-(3-methylphenoxymethyl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indazole
1-[2-(3-methoxyphenyl)-1,3-benzoxazole-6-carbonyl]-N,N-dimethylpyrrolidin-3-amine
3-(2-methoxy-6-methylphenyl)-1-(oxan-4-ylmethyl)urea
3-[4-(dimethylamino)phenyl]-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]propan-1-one
N,N-diethyl-2-{[2-oxo-4-(oxolane-3-carbonyl)-1-(2-phenylethyl)-1,4-diazepan-6-yl]oxy}acetamide
3-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1R,5R)-3-(4-chloro-2-methylbenzoyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-(2-phenoxyethyl)-1,4-diazepan-5-one
methyl 6-(2-{[(dimethyl-1,3-thiazol-5-yl)formamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)pyridine-3-carboxylate
N-methyl-2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]acetamide
N-[(3S,4R)-1-(4-cyanopyridin-2-yl)-4-propylpyrrolidin-3-yl]acetamide
(3S)-4-{2-[(3-chlorophenyl)methyl]-1,3-benzoxazole-6-carbonyl}-1,3-dimethylpiperazin-2-one
5-methyl-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(4-hydroxyazepan-4-yl)methyl]-2,3-dihydro-1,4-benzodioxine-6-sulfonamide
5-(1-benzofuran-2-yl)-2-methyl-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
4-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}pyrimidin-2-amine
1-[7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
2-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-N-propylacetamide
N-(3-{4-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}phenyl)pyridine-4-carboxamide
(3R,4S)-1-[(5-methylpyrazin-2-yl)methyl]-4-propylpyrrolidin-3-amine
1-[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(methylsulfanyl)ethan-1-one
2-methyl-4-[4-(piperidin-1-yl)piperidin-1-yl]-6-(propan-2-yl)pyrimidine
2-(cyclopropylmethyl)-9-(2-hydroxy-4-methoxybenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}[(4-fluorophenyl)methyl]methylamine
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-2-methylpropanamide
5-(azepan-1-yl)-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(1H-indol-2-ylmethyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-3-ol
N-butyl-3-{[4-(3-methoxyphenyl)piperazin-1-yl]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
methyl[(1-methyl-1H-pyrazol-4-yl)methyl]{[2-(trifluoromethyl)phenyl]methyl}amine
(2H-1,3-benzodioxol-4-ylmethyl)[(4-fluorophenyl)methyl](pyridin-4-ylmethyl)amine
1-[2-(methylsulfanyl)benzoyl]-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
N-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]acetamide
N-methyl-2-(2-methylphenyl)-N-(quinolin-8-ylmethyl)benzamide
(2R,3R)-3-[ethyl(methyl)amino]-1'-(4-methylpyrimidine-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(1S,5R)-N-(naphthalen-1-yl)-10-oxo-3,9-diazabicyclo[3.3.2]decane-3-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}ethan-1-ol
4-(3-hydroxy-3-methylbutyl)-N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]benzamide
2-[1-(thiophen-3-yl)propan-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(2-fluorophenyl)methyl]-3-[1-(3-phenylprop-2-ynoyl)piperidin-3-yl]propanamide
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}[(2E)-3-(furan-2-yl)prop-2-en-1-yl]methylamine
2,3,6-trimethyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]quinoline-4-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
ethyl 4-[1-(furan-3-ylmethyl)piperidin-3-yl]piperazine-1-carboxylate
1-(carbamoylmethyl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]piperidine-4-carboxamide