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4-{[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1-methyl-1H-pyrazole
N-[(3R,4S)-4-cyclopropyl-1-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
3-[(3R,4S)-1-[(3-methylphenyl)carbamoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
2-{4-[(2-phenoxyethyl)amino]piperidin-1-yl}pyridine-4-carbonitrile
3-({[1-(2-chloro-6-methylbenzoyl)piperidin-4-yl]oxy}methyl)pyridine
3-(3-fluorophenyl)-6-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(oxan-4-yl)ethyl]amine
(isoquinolin-5-ylmethyl)(methyl){[3-(morpholin-4-ylmethyl)phenyl]methyl}amine
5-({4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-2-(pyridin-2-yl)pyrimidine
2-(pyridin-2-yl)-5-{1-[3-(pyridin-4-yl)propyl]-1H-imidazol-2-yl}pyrimidine
N-[4-(2-fluorophenoxy)phenyl]-1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidine-4-carboxamide
2-(4-chlorophenyl)-4-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}morpholine
4-(2-phenylphenyl)-3-[2-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[4-(4-{[3-(1H-1,2,3-benzotriazol-1-yl)propyl]amino}piperidin-1-yl)phenyl]cyclopentanecarboxamide
(2S,4S,5R)-4-[(cyclopent-3-en-1-yl)carbamoyl]-2-ethyl-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
5-[(4-acetamidophenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(3-methylpyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-(3-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-3-oxopropyl)-5-[(4-methylphenyl)methyl]pyrrolidin-2-one
4-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-7-(3-chlorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-(methoxymethyl)-1-methyl-N-[(4-phenyloxan-4-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3aS,7aR)-2-(2,5-dimethyl-1-phenyl-1H-pyrrole-3-carbonyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-(thiophen-3-ylmethyl)benzamide
ethyl 4-[2-(phenylamino)pyrimidine-5-carbonyl]piperazine-1-carboxylate
4-(1-benzyl-1H-imidazol-2-yl)-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidine
4-benzyl-2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
(4aR,8aR)-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-octahydro-2H-1,4-benzoxazine
1-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
2-{4-[6-amino-5-cyano-4-(5-cyano-1-methyl-1H-pyrrol-3-yl)pyridin-2-yl]phenoxy}acetic acid
4-[(3-phenyl-1H-pyrazol-5-yl)methyl]-4H-1,2,4-triazole
(4aR,8aR)-7-(6-cyanopyridin-2-yl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
1-{3-[4-(2-methoxyphenoxy)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
N-[(5-chlorothiophen-2-yl)methyl]-1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
6-cyclopentyl-1-methyl-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{6-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]pyridin-2-yl}ethan-1-ol
N-[3-(dimethylamino)-2,2-dimethylpropyl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(propan-2-yl)-3-(pyridin-3-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanamide
1-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine
{[3-(benzyloxy)phenyl]methyl}[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
5,6-dimethyl-2-oxo-N-[(2-phenoxypyridin-3-yl)methyl]-1,2-dihydropyridine-3-carboxamide
1-methyl-N-(6-methylpyridin-3-yl)-6-oxopiperidine-3-carboxamide
2-methoxy-4-{[2-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1H-imidazol-1-yl]methyl}phenol
4-methoxy-3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-methylbenzamide
2-(2-{[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]amino}ethyl)-6-methyl-3,4-dihydropyrimidin-4-one
7-(4-fluorophenyl)-2-{2-[(pyridin-3-yl)amino]ethyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(2S,4S)-4-amino-1-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazole-5-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
5-(2,6-dimethoxyphenyl)-3-(3-propoxypiperidin-1-yl)-1,2,4-triazine
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]butan-1-one
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N,N-bis(prop-2-en-1-yl)benzamide
3-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-1-(2-hydroxypyridin-3-yl)urea