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6-(2,5-dimethoxyphenyl)-2-(morpholin-4-yl)pyrimidin-4-amine
1-[1-(2,5-difluorobenzoyl)piperidin-4-yl]-2-phenylethan-1-ol
5-chloro-4-methyl-6-(4-{[2-(morpholin-4-yl)ethyl]amino}piperidin-1-yl)pyrimidin-2-amine
1-[2-(furan-2-yl)azepan-1-yl]-2-(3-hydroxyphenyl)ethan-1-one
(1R,5S,8S)-8-hydroxy-N-{4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}-3-azabicyclo[3.2.1]octane-3-carboxamide
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-(3-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]methyl}phenyl)ethan-1-one
3-[(3R,4S)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
2-[methyl(pyridin-2-ylmethyl)amino]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(1R,5R)-N-(2,3-dichlorophenyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-(thiomorpholin-4-yl)-2-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}morpholin-3-yl)ethan-1-one
4-({1-[(2S)-2-aminopropanoyl]piperidin-4-yl}oxy)-3-chloro-N-cyclopentylbenzamide
5-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4-phenylpyrimidin-2-amine
2-(dimethylamino)-2-(3-fluorophenyl)-1-[4-(thian-4-yl)piperazin-1-yl]ethan-1-one
N-cyclopropyl-N-{[1-(3-phenoxypropyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}acetamide
4-(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)phenol
(3S,4R)-1-(dimethyl-1,3-thiazole-5-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
{1-[({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)methyl]cyclobutyl}methanol
1-methyl-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1H-pyrazole-5-carboxamide
N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-4-sulfamoylbenzamide
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-(1H-pyrazol-1-yl)butanamide
N,N-dimethyl-2-[4-(piperidine-1-carbonyl)pyridin-2-yl]aniline
N-{3-[1-(2-methylpyridin-4-yl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]propyl}acetamide
4-methoxy-3-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}benzene-1-sulfonamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-3-yl]-5-methylpyrazine-2-carboxamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(pyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-(5-methylpyrazin-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-{5-[4-phenyl-1-(pyridin-3-ylmethyl)-1H-imidazol-5-yl]thiophen-2-yl}prop-2-yn-1-ol
[3-(cyclopropylmethyl)-1-[2-(diethylamino)ethyl]piperidin-3-yl]methanol
1-[1-(5-butyl-4-phenyl-1H-imidazol-1-yl)butan-2-yl]-4-methylpiperazine
8-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-8-azaspiro[4.5]decane-7,9-dione
2-[(dimethylcarbamoyl)amino]-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)acetamide
2-cyclopropyl-N-[1-(methylcarbamoyl)cyclohexyl]pyrimidine-5-carboxamide
(3R,5S)-1-benzyl-N-cyclopentyl-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(trimethylpyrimidin-4-yl)pyrrolidin-3-yl]methanol
1-(propan-2-yl)-4-{4-[2-(pyridin-2-yl)ethyl]piperazine-1-carbonyl}pyrrolidin-2-one
2-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-(2-hydroxy-3-{2-[(3-hydroxyazetidin-1-yl)methyl]-4-methoxyphenoxy}propyl)piperidin-4-ol
(2S)-1-({1-[1-(2-methylpyridin-4-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)pyrrolidine-2-carboxamide
1-[(2-phenyl-1,3-thiazol-5-yl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
5-{[(1S,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-2,1,3-benzothiadiazole
3,5-dimethoxy-2-({methyl[(1-methylpiperidin-2-yl)methyl]amino}methyl)benzoic acid
(2S)-1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-hydroxy-2-phenylethan-1-one
1-{4-[1-(3-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-4-oxobutyl}pyrrolidin-2-one
ethyl 3-benzyl-1-[(2-methylphenyl)carbamoyl]piperidine-3-carboxylate
N-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-3-(1,2-oxazinan-2-yl)propanamide
[1-(2-methanesulfonylethyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
2-methyl-5-(2-methyl-1H-imidazol-4-yl)quinoline
1,6-dimethyl-3-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
3-(1-methyl-1H-pyrrol-2-yl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1H-pyrazole-5-carboxamide