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1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3-(3-methoxyphenoxymethyl)piperidine
1-(2-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidine-1-carbonyl}phenyl)ethan-1-one
(1S,5R)-1,3,3-trimethyl-6-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]-6-azabicyclo[3.2.1]octane
1-[1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]piperidin-3-ol
2-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}-6,8-dimethylquinolin-4-ol
N-[(2S)-1-[3-(3-methoxyphenoxy)azetidin-1-yl]-4-methyl-1-oxopentan-2-yl]acetamide
2-methanesulfonyl-N-methyl-N-[1-(pyridin-3-yl)ethyl]acetamide
3-(4-methoxyphenoxymethyl)-1-(1H-pyrrole-3-carbonyl)piperidine
2-[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]-1-(1,4-dioxan-2-ylmethyl)-1H-imidazole
2-(carbamoylamino)-N-[(4-fluorophenyl)(pyridin-4-yl)methyl]acetamide
(3R,5R)-N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
4-{3-[4-(pyrazin-2-yl)piperazine-1-carbonyl]phenyl}morpholine
1-(2-{4-[(benzylamino)methyl]-3-methyl-1H-pyrazol-1-yl}ethyl)piperidine-4-carbonitrile
2,6-dimethyl-4-(1-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-imidazol-2-yl)phenol
N'-ethyl-N'-[2-(morpholin-4-yl)ethyl]ethanediamide
N-cycloheptyl-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
7-chloro-N,3,5-trimethyl-N-(pyrazin-2-ylmethyl)-1-benzofuran-2-carboxamide
2-{1-[(2-fluorophenyl)methyl]-4-[(2,3,6-trifluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
3-{1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-4-yl}phenol
N-(4-chloro-3-methylphenyl)-2-{[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](propan-2-yl)amino}acetamide
(2R,6S)-4-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,6-dimethylmorpholine
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)[(8-fluoroquinolin-2-yl)methyl](2-methoxyethyl)amine
[3-(1,3-benzoxazol-2-yl)propyl](benzylsulfamoyl)amine
2-hydroxy-1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
N-[2-(methylsulfanyl)phenyl]-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)cyclopropanecarboxamide
1-cyclopentyl-N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
N-{2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}-2-(4-phenylphenyl)acetamide
N-[2-(3-chlorophenyl)ethyl]-1-(2-methoxyethyl)-5-(2-methylpiperidine-1-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[(1s,4s)-4-aminocyclohexyl]-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-1H-1,2,3-triazole-4-carboxamide
3-(prop-2-en-1-yl)-1-[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperidine-3-carboxylic acid
[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl](methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]benzamide
2-(2-methyl-1,3-thiazol-4-yl)-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
2-(3-hydroxypropyl)-9-[(4-methylnaphthalen-1-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[(5-methylpyrazin-2-yl)methyl]acetamide
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-(thian-4-yl)acetamide
4-{4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]phenyl}-4H-1,2,4-triazole
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-2,2-diphenylacetamide
1-(2-methylphenyl)-4-{1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-3-yl}piperazine
1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(2-methoxyethoxy)piperidine
4-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]-8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(3R,4R)-3-hydroxy-1-[2-(2-oxopiperidin-1-yl)acetyl]piperidin-4-yl]pyrazine-2-carboxamide
N-[2-(pyridin-2-yl)ethyl]-6-[3-(trifluoromethyl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
6-(2,4-difluoro-3-methoxybenzoyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
(3aR,6aR)-2-[6-methyl-2-(morpholin-4-yl)pyrimidin-4-yl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{3-oxo-3-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]propyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(3-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-3-oxopropyl)pyrrolidin-2-one
2-(2H-1,3-benzodioxol-5-yl)-2-(4-methyl-1,4-diazepan-1-yl)acetic acid
(3R,5R)-5-(morpholine-4-carbonyl)-N-[2-(phenylsulfanyl)ethyl]piperidine-3-carboxamide