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N-[(2-chlorophenyl)methyl]-3-{1-[3-(methylsulfanyl)propanoyl]piperidin-3-yl}propanamide
2-methanesulfonyl-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)acetamide
1-benzyl-5-[(3-hydroxyphenyl)methyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[2-(morpholin-4-yl)ethyl]-5-[4-(pyridin-4-yl)piperidine-1-carbonyl]piperidin-2-one
(1R,2R,6S,7S)-4-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
2-({3-cyclopentyl-1-[(2-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)-5,6-dimethyl-2,3-dihydropyridazin-3-one
2-{4-[1-(2H-1,3-benzodioxol-4-ylmethyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
7-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazine-1-carbonyl]thiophene-3-sulfonamide
2-(ethylamino)-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}pyrimidine-5-carboxamide
N,N-diethyl-4-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]aniline
methyl[(4-{[1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl](2-phenylethyl)amine
3-{2-oxo-2-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}imidazolidine-2,4-dione
4-(5-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
(benzylsulfamoyl)[(2-methylphenyl)(pyridin-4-yl)methyl]amine
7-methyl-4-{2-oxo-2-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethyl}-2H-chromen-2-one
2-{4-[(4Z)-hept-4-en-1-yl]piperazin-1-yl}-5-methylpyrimidin-4-amine
1-[3-(3-benzoylpiperidin-1-yl)-3-oxopropyl]-1,2-dihydropyridin-2-one
N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
3-[3-(hydroxymethyl)phenyl]-5-[(propan-2-yl)sulfamoyl]benzoic acid
(3R,4R)-3-(hydroxymethyl)-N,N-dimethyl-4-(morpholin-4-ylmethyl)pyrrolidine-1-sulfonamide
1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(dimethylamino)propan-1-one
N-{[3-(methylsulfanyl)phenyl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-(naphthalen-1-ylmethyl)-3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]piperazin-2-one
1-(adamantan-1-yl)-4-(5-methyl-1,3-oxazole-4-carbonyl)piperazine
3-{[(cyclopropylmethyl)(2-methoxyethyl)amino]methyl}-6-methyl-1,2-dihydroquinolin-2-one
N-[(4-methoxynaphthalen-1-yl)methyl]-3-(4-methylpiperazin-1-yl)-N-(propan-2-yl)propanamide
1-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-phenoxyethan-1-one
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanamide
N-[(3-{1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)methyl]propanamide
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl){[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
(1R,5S)-3-[(2,3-dichlorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(1,3-benzothiazol-2-yl)-N-[(4-hydroxyazepan-4-yl)methyl]propanamide
2-(2-{5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoethyl)-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
1-(3-{[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]methyl}phenyl)ethan-1-one
5-methanesulfonyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-4-(piperidin-3-yl)pyrimidin-2-amine
1-[4-(3-chlorophenyl)phenyl]-3,3-bis(2-methoxyethyl)urea
1-[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]azepane
7-(ethanesulfonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-fluoro-2-{1-[3-(1H-1,2,4-triazol-1-yl)propyl]piperidin-2-yl}-1H-1,3-benzodiazole
1-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
1-[2-(morpholin-4-yl)benzoyl]azepan-3-amine
N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]furan-2-carboxamide
{1-[1-(6-ethoxy-4-methylquinazolin-2-yl)piperidine-4-carbonyl]piperidin-4-yl}(pyridin-3-yl)methanol
1-[2-(3-chloro-5-fluoro-4-methoxyphenyl)-1H-imidazol-1-yl]propan-2-ol
5-methoxy-2-{[2-(trifluoromethyl)morpholin-4-yl]methyl}-4H-pyran-4-one
3-{2-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}phenol
4-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-1-methyl-2-phenylpiperazine
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}oxolane-2-carboxamide
1-(propan-2-yl)-4-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}-1,4-diazepane