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N-cyclopropyl-1-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
N-(2-oxopyrrolidin-3-yl)-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-3-(1,2-oxazinan-2-yl)propanamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(diethylamino)methyl]phenoxy]-N-(5-fluoro-2-methylphenyl)acetamide
8-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
1-[2-hydroxy-3-(4-{[(2-hydroxyethyl)(methyl)amino]methyl}-2-methoxyphenoxy)propyl]piperidin-4-ol
2-{5-[2-(5-methyl-1H-pyrazol-1-yl)ethyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}pyridine
1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
1-(azepan-1-yl)-3-[3-({[2-methyl-2-(morpholin-4-yl)propyl]amino}methyl)phenoxy]propan-2-ol
N-(2,4-dimethoxyphenyl)-3-{1-[3-(pyridin-4-yl)propanoyl]piperidin-4-yl}propanamide
3-{[5-(pentan-3-yl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]methyl}pyridine
4-[2-(3-methylbut-2-en-1-yl)-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl]benzonitrile
1-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-2-(2-methoxyphenyl)pyrrolidine
N2-(2-methoxyethyl)-N4-methyl-N4-(1,3-thiazol-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
dimethyl(2-{5-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,2,4-oxadiazol-3-yl}ethyl)amine
ethyl 4-{[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]amino}piperidine-1-carboxylate
2-(3-chloro-4-hydroxyphenyl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
4-({2-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
5-methoxy-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N,1-dimethyl-1H-indole-2-carboxamide
3-[1-(3-methylfuran-2-carbonyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
7-(4-chlorophenyl)-2-(1H-imidazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[(1-ethyl-1H-indol-3-yl)sulfanyl]-1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]ethan-1-one
methyl 4-[2-(cyclohexylmethyl)morpholin-4-yl]-4-oxobutanoate
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
2-[(4aR,7aS)-6,6-dioxo-4-(1,3-thiazol-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
N-methyl-N-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]oxan-4-amine
3-(4-chlorophenyl)-2-{4-[5-(hydroxymethyl)furan-2-yl]-1H-1,2,3-triazol-1-yl}propan-1-ol
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-4-methoxybenzamide
6-[(diethylamino)methyl]-N-(2-phenylpropyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-2-(4-methoxyphenyl)ethan-1-one
N-(3-chloro-4-methoxyphenyl)-3-[1-(4-phenylbutanoyl)piperidin-3-yl]propanamide
5-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole
3-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-1,2-oxazole-5-carboxamide
1'-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(adamantan-2-ylmethyl)-1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-amine
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-ethyl-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
(3R,4R)-1-(2-methyl-5-propylpyrimidin-4-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-ol
4-[4-(1-benzylpiperidin-4-yl)piperazin-1-yl]-2-[(3,4-dimethoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
(benzylsulfamoyl)[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
4-(4,4-difluoropiperidine-1-carbonyl)-7-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
8-benzyl-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[2-(2-fluorophenyl)acetyl]-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-methyl-2-(methylsulfanyl)-N-[1-(pyridin-2-yl)propan-2-yl]pyridine-3-carboxamide
3-({[(1-benzyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)pyrrolidin-3-ol
{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}({[2-(morpholin-4-yl)pyridin-3-yl]methyl})amine
2-(2-oxo-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-2-azaspiro[4.5]decan-3-one
2-cyclopentyl-1-[4-(3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]ethan-1-one
7-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}quinolin-8-ol