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4-(5-methylpyridin-2-yl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidin-4-ol
2-(cyclopropylmethyl)-7-[2-(methylamino)pyridine-4-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl({[5-(oxan-2-yl)thiophen-2-yl]methyl}){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
3-chloro-4-({4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)phenol
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
4-{1-[2-(3-methylphenyl)benzoyl]piperidin-4-yl}morpholine
methyl({[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}){[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
2,3,5-trimethyl-N-[2-(morpholin-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-{1-[(2E)-3-(2-fluorophenyl)prop-2-enoyl]piperidin-3-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
6-{2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-3-carbonitrile
7-(2-methylphenyl)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-cyclopropyl-2-(3-{[methyl({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-2-methanesulfonamidoacetamide
4-[1-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)piperidin-4-yl]thiomorpholine
4-[4-(naphthalen-1-ylmethyl)piperazin-1-yl]-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
methyl 5-(cyclopentylamino)-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{2-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}-1-methyl-1H-1,3-benzodiazole
methyl 5-[(1-hydroxypropan-2-yl)amino]-3-(oxolane-2-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
methyl({[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl})(1,3-thiazol-2-ylmethyl)amine
6-{[3-(hydroxymethyl)morpholin-4-yl]methyl}pyridine-2-carboxylic acid
methyl 6-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)-3-(oxolane-2-amido)thieno[2,3-b]pyridine-2-carboxylate
1-(1,3-benzothiazole-6-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
4-(4-{[4-(1-methoxypropan-2-yl)piperidin-1-yl]methyl}phenyl)-2-methylbutan-2-ol
2-methyl-3-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydroisoquinoline
N,N-dimethyl-4-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]benzene-1-sulfonamide
3-[(2R,3R,6R)-5-(4-methyl-1H-imidazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
5,6-dimethyl-3-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-1,2-dihydropyridin-2-one
methyl 5-(2,6-dimethylquinoline-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}oxolane-3-carboxamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-methyl-N-(1,3-thiazol-2-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
N-[2-(azepan-1-yl)ethyl]-N-ethyl-2-methyl-5-sulfamoylbenzamide
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-1-methyl-1H-pyrazole-5-carboxamide
N-(1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
3-amino-1-{[4-methoxy-3-(prop-2-en-1-yl)phenyl]methyl}pyrrolidine-3-carboxylic acid
methyl 8-(9H-fluoren-2-ylmethyl)-1-methoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2-({[(3R,4R)-1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
(4aS,7aR)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(cyclohexylmethyl)-5-[(5-hydroxyadamantan-2-yl)amino]-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-cyclopentyl-4-{4-[4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}pyrrolidin-2-one
4-[1-(1-{[3-(4-chlorophenoxy)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carbonyl]morpholine
N-(1-{7-[(2-hydroxy-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-5-(methoxymethyl)furan-2-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3-{[(3R)-3-hydroxypyrrolidin-1-yl]sulfonyl}benzamide
2-(2-methylphenyl)-6-(4H-1,2,4-triazol-4-yl)-1,3-benzoxazole
7-[cyclohexyl(methoxy)methyl]-4-(oxolane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]-2-(4-propanoylphenoxy)acetamide
2-cyclopropyl-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-imidazole
3-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]benzonitrile
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-4-methoxy-N-(pyridin-4-ylmethyl)benzamide
3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(5-fluoro-2-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one