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(2H-1,3-benzodioxol-5-ylmethyl)(methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
(1S,5R)-6-[(2-fluoro-5-methoxyphenyl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
cyclopentyl 4-{[(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)carbamoyl]amino}benzoate
7-{3-[hydroxy(phenyl)methyl]-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl}-1,2,3,4-tetrahydroquinoxalin-2-one
2-{1-[(2-ethoxyphenyl)methyl]-4-[(3-methyl-1H-indol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
5-({[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}sulfanyl)-1H-1,2,4-triazol-3-amine
3-(4-fluorophenyl)-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-2-methoxy-N,4-dimethyl-1,3-thiazole-5-carboxamide
3-[3-(2-phenylacetyl)piperidine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
N-[(3S,4R)-1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
2-methyl-3-{[2-(1,3-thiazol-2-yl)piperidin-1-yl]methyl}quinoxaline
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-chloro-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]benzamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-(4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-1-(1-methylpiperidin-4-yl)piperazin-2-yl)ethan-1-ol
N-[2-(dimethylamino)-2-(4-methylphenyl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
1-{4-[(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)amino]piperidin-1-yl}ethan-1-one
7-methoxy-4-methyl-2-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}quinazoline
N-(2,2-dimethyloxan-4-yl)-5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carboxamide
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(cyclopent-1-ene-1-carbonyl)-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
ethyl 3-[(2-fluorophenyl)methyl]-1-(pyridine-3-carbonyl)piperidine-3-carboxylate
2-methyl-6-[5-(oxan-4-yl)-4-phenyl-1H-imidazol-1-yl]heptan-2-ol
N-[(1R)-2,3-dihydro-1H-inden-1-yl]-6-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
1-(2-cyclohexylethyl)-3-({[(4-fluorophenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
2-{3-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]piperidin-1-yl}acetamide
1-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]-2-(2,3,4-trifluorophenyl)ethan-1-one
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-4-methoxybenzamide
1-ethyl-3-[1-(2-phenoxyethyl)-1H-imidazol-2-yl]piperidine
1'-(3-fluoropyridin-2-yl)-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}acetamide
6-chloro-3-{[1-(hydroxymethyl)cyclobutyl]methyl}-8-methyl-3,4-dihydroquinazolin-4-one
2-(4-chlorophenyl)-4-(3-propyl-1H-pyrazole-4-carbonyl)morpholine
2-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}-1-methyl-1H-indole
4-({9-oxo-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-2-yl}methyl)benzonitrile
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-5-(4-methoxyphenyl)furan-2-carboxamide
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1,3-benzothiazole-6-carboxamide
1-(4-fluorophenyl)-4-[1-(thian-4-yl)piperidin-3-yl]piperazine
N-(furan-2-ylmethyl)-N-{[2-(4-methoxyphenyl)-8-methylquinolin-3-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
7-fluoro-2-methyl-4-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}quinoline
2-{1-[(4-fluorophenyl)methyl]-4-(thian-4-yl)piperazin-2-yl}ethan-1-ol
N-(2-{[(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]piperidin-3-yl]formamido}ethyl)acetamide
N,N-dimethyl-2-[(1S,5R)-6-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
1-ethyl-3-methyl-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}piperidine-3-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(1-cyclopropyl-6-oxopiperidine-3-carbonyl)piperazin-2-one
(2R,6S)-4-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-2,6-dimethylmorpholine
2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)-N-{[3-(trifluoromethoxy)phenyl]methyl}acetamide
7-(1,3-benzothiazol-2-yl)-4-(3-phenylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{5-[2-(diethylamino)ethyl]-1,3,4-thiadiazol-2-yl}-2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carboxamide
N,1-dimethyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine