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N-cyclopentyl-1,3-dimethyl-N-({3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-1H-pyrazole-5-carboxamide
1-[(4-fluorophenyl)methyl]-4-(5-methyl-1,3-oxazole-4-carbonyl)-2-(propan-2-yl)-1,4-diazepane
1-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(2-methylphenyl)piperazine
4-(2-ethoxyphenyl)-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
2-(4-chloro-2-methylphenoxy)-1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]ethan-1-one
1-ethyl-2-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}methyl)-1H-1,3-benzodiazole
N-(1-benzothiophen-5-ylmethyl)-2-(piperazin-1-yl)acetamide
(4aS,8aR)-1-(3-aminopropyl)-6-(1H-imidazol-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
N-(2-hydroxy-2-phenylethyl)-2-(3-methoxyphenyl)-N-methyl-1,3-benzoxazole-6-carboxamide
5,6-dimethyl-3-[3-(naphthalene-1-carbonyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
N4-ethyl-N2-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-N4-methylpyrimidine-2,4-diamine
3-methyl-4-(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)piperazin-2-one
4-benzyl-5-[(3-methylthiophen-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-(1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-4-yl)-2-phenylethan-1-ol
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}[(5-ethylpyridin-2-yl)methyl]amine
4-(3-{[3-(dimethylamino)propyl](methyl)amino}piperidine-1-carbonyl)-2-methoxyphenol
4-methoxy-N-{1-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
1-ethyl-4-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridin-2-one
N-[2-(furan-2-yl)-2-hydroxyethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-(6-methoxy-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-2-(pyridin-3-yl)piperidine-1-carboxamide
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-[2-(pyridin-2-yl)ethyl]-1,4-diazepan-5-one
1-cyclopentyl-N-[2-methyl-2-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
N-cyclopropyl-4-methoxy-2-{[1-(pyrimidin-2-yl)piperidin-4-yl]oxy}benzamide
2-[2-({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
(2S,4S)-1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-4-cyclopropaneamido-N-ethylpyrrolidine-2-carboxamide
7-(oxane-4-carbonyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(4-{1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-phenyl-1H-imidazol-5-yl}phenyl)prop-2-yn-1-ol
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-5,6-dimethylpyridine-3-carboxamide
(1-{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-4-yl)methanol
2-(4-fluorophenoxymethyl)-N-methyl-N-(oxan-2-ylmethyl)-1,3-oxazole-4-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
N-methyl-N-{2-phenyl-1-[1-(thiolan-3-yl)piperidin-4-yl]ethyl}thiophene-3-carboxamide
2-[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]-2,8-diazaspiro[4.5]decane
N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-1,3-benzothiazole-6-carboxamide
4-[4-(2-chlorophenoxy)piperidine-1-carbonyl]benzonitrile
1-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
2-(3-hydroxyphenyl)-2-{methyl[4-(morpholin-4-yl)butyl]amino}acetic acid
5-(2-methylphenyl)-N-[2-(pyrazin-2-yl)ethyl]-1,2,4-triazin-3-amine
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[4-(trifluoromethyl)benzoyl]piperidine
6-methyl-5-(4-methyl-1H-pyrazol-1-yl)pyridin-2-amine
5-ethyl-1'-(quinoline-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[(4-fluorophenyl)formamido]-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methylpropanamide
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(2-propoxyacetyl)-1,4-diazepan-5-one
2-[4-(hydroxymethyl)-4-[(4-methoxyphenyl)methyl]piperidin-1-yl]pyridine-4-carbonitrile
N,N-dimethyl-2-{4-[3-methyl-5-(phenoxymethyl)furan-2-carbonyl]morpholin-3-yl}acetamide
3-(4-methyl-1,3-thiazol-5-yl)-1-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
3-(2-{[(3-methoxyphenyl)methyl]carbamoyl}ethyl)-N-[4-(methylsulfanyl)phenyl]piperidine-1-carboxamide
N-cyclopropyl-2-{[3-(3-hydroxy-3-methylbutyl)phenyl]formamido}acetamide