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1-(3-methyl-1H-pyrazole-5-carbonyl)-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
(2S,4S)-1-{[4-(benzyloxy)phenyl]methyl}-N-[(4-methylphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[1-ethyl-3-(hydroxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
5-fluoro-2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-3-methyl-1H-indole
3-[({1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}oxy)methyl]pyridine
5-(4-ethylphenyl)-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-[(4-methylphenyl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
9-(but-3-yn-1-yloxy)-4-cyclohexanecarbonyl-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-(1,2-oxazolidin-2-ylmethyl)piperidin-2-one
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-[3-(propan-2-yl)adamantan-1-yl]urea
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-[3-(methylsulfanyl)butyl]cyclopropanamine
N-{[5-(1-benzofuran-5-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-methoxyacetamide
1-(3-fluoro-5-methylphenyl)-3-(5-hydroxypentyl)urea
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-acetamido-N-(pyridin-3-ylmethyl)propanamide
(1S,8R)-4-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-3-azatricyclo[6.2.1.02,7]undeca-2,4,6-triene-5-carbonitrile
2-{[(2-methoxyethyl)(1-methylpiperidin-4-yl)amino]methyl}-5,8-dimethylquinolin-4-ol
{1-[(4-chlorophenyl)methyl]-3-(2-phenoxyethyl)piperidin-3-yl}methanol
4-[1-(3,5-difluoro-4-methoxybenzoyl)pyrrolidin-3-yl]benzoic acid
1-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
5-methoxy-3-[1-(pyridin-3-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
(1S,4S)-2-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,5-diazabicyclo[2.2.1]heptane
{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-2,5-dihydro-1H-pyrrol-2-yl}methanol
1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)butan-1-one
3-(pyrrolidine-1-carbonyl)-1-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]piperidine
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-[3-(pyridin-3-yl)propyl]-1H-pyrazole-4-carboxamide
1-[(4-methoxyphenyl)methyl]-4-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-4-phenylbutane-1,4-dione
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-2,3-dimethoxybenzamide
2-(5-acetylthiophen-3-yl)-N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
ethyl 1-[(4-hydroxy-2-methoxyphenyl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
2-ethyl-4-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}pyrimidine
3-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-3-yl}-N-(4-fluoro-2-methylphenyl)propanamide
(2R,3R,6R)-3-phenyl-5-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2,6-dimethoxybenzamide
1-(furan-2-carbonyl)-4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazine
3-fluoro-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyridine-4-carboxamide
8-(2,1,3-benzoxadiazol-5-ylmethyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-(pentan-2-yl)-8-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-methyl-7-(6-methylpyridazin-3-yl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]-2-(1H-pyrazol-1-yl)benzamide
7-[(4-phenylpiperazin-1-yl)methyl]-4-(2,4,5-trifluorobenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-methyl-N-{2-[2-(methylcarbamoyl)ethyl]phenyl}-4-(2-methylpropyl)-3-oxopiperazine-1-carboxamide
N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-2-(4-phenylpiperidin-1-yl)acetamide
N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
methyl 3-(cyclobutylmethoxy)-5-[(1S,4S)-5-methyl-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]benzoate
8-(4-chloro-3-methylbenzoyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]phenol
dimethyl({2-[4-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenoxy]ethyl})amine
2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[2-(methylsulfamoyl)ethyl]acetamide