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6-(4-fluorophenyl)-2-[(3R)-3-hydroxypyrrolidine-1-carbonyl]-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-[(4-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-methoxyphenyl)-1-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}propan-2-ol
2-[2-(4-ethylpiperazin-1-yl)ethyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(furan-2-yl)-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}-N-[(4-chlorophenyl)methyl]piperidine-1-carboxamide
2-(azepane-1-carbonyl)-6-(2-chlorophenyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
2-(4-fluorophenoxymethyl)-N-(oxan-2-ylmethyl)-1,3-oxazole-4-carboxamide
(4aS,7aR)-1-(3-hydroxy-4-methylbenzoyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[3-(2-methoxyphenyl)propyl]piperidin-3-amine
3-(4-chlorophenyl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]-3-phenylpropanamide
2-[methyl(pyridin-4-ylmethyl)amino]-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
1-(2-methoxyethyl)-8-[(1-methyl-1H-indol-3-yl)methyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(azepane-1-carbonyl)-1-(butan-2-yl)-4-oxo-N-(3-phenylpropyl)-1,4-dihydropyridine-3-carboxamide
3-(azocan-1-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]propanamide
3-[1-(1-cyclopentanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-1-(2-methoxyphenyl)urea
1-(4,6-dimethoxypyrimidin-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-[1-(4,4,4-trifluorobutyl)pyrrolidin-3-yl]benzoic acid
N-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-5-methyl-N-(pyridin-3-ylmethyl)thiophene-2-carboxamide
[2-({4-[(3-chloro-2,6-difluorophenyl)methyl]piperazin-1-yl}methyl)phenyl]methanol
1-(1,2,3-thiadiazole-4-carbonyl)-3-[4-(trifluoromethyl)benzoyl]piperidine
(2S)-2-amino-1-[5-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]pentan-1-one
2-amino-6-(3,5-difluorophenyl)-4-(3,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
(2S,4S)-1-[(2E)-but-2-en-1-yl]-N-ethyl-4-(7-methyl-1-benzofuran-2-amido)pyrrolidine-2-carboxamide
5-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}-N,N-dimethylpyridin-2-amine
N-cyclohexyl-N,5-dimethyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
1-cyclopropyl-4-{7,7-dimethyl-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}pyrrolidin-2-one
1-(4-methylphenyl)-4-[2-(4-methylphenyl)acetyl]piperazin-2-one
N-[2-({2-oxo-2-[3-oxo-2-(propan-2-yl)piperazin-1-yl]ethyl}sulfanyl)phenyl]acetamide
2-methoxyethyl 2-(pyridin-2-yl)piperidine-1-carboxylate
N,6-dimethyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-N-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-[methyl(pyridin-3-ylmethyl)amino]-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]acetamide
(2S)-2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]propanamide
3-({ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-7-methoxy-1,2-dihydroquinolin-2-one
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)acetamide
2-({[(1S,2R)-2-(hydroxymethyl)cyclopentyl]amino}methyl)-5,8-dimethylquinolin-4-ol
(1s,4s)-4-{[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}cyclohexan-1-amine
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carboxamide
N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-[4-(pyridin-2-yl)-1H-pyrazol-1-yl]acetamide
4-methoxy-3-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}benzamide
(3ar,6ar)-N-[(3-hydroxyphenyl)methyl]-N-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-[4-(1H-indol-2-ylmethyl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
1-[benzyl(methyl)amino]-3-[4-(1,4-oxazepan-4-ylmethyl)phenoxy]propan-2-ol
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-[3-(2-methylphenyl)-1H-pyrazol-1-yl]acetamide
4-(hydroxymethyl)-3-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1,3-oxazolidin-2-one
(3S,4S)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-(1H-imidazol-2-yl)pyrrolidine-3-carboxylic acid
(1-benzothiophen-2-ylmethyl)(methyl)[(4-{2-[4-(pyridine-4-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amine
7-(1-phenylcyclohexanecarbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
4-{2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-oxoethyl}-1λ6-thiane-1,1-dione
4-[(2,5-difluorophenyl)methyl]-9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine